All Stories

  1. Effects of orexin receptor antagonism on human sleep architecture: A systematic review
  2. Circadian disruption impairs fear extinction and memory of conditioned safety in mice
  3. The Killing Mechanism of Teixobactin against Methicillin-Resistant Staphylococcus aureus: an Untargeted Metabolomics Study
  4. Long-term Outcomes After Controlled Oxygenated Rewarming of Human Livers Before Transplantation
  5. SMAD4 protein is decreased in the dorsolateral prefrontal and anterior cingulate cortices in schizophrenia
  6. Curcumin Attenuates Colistin-Induced Peripheral Neurotoxicity in Mice
  7. Hypnotics with novel modes of action
  8. Separating Probability and Reversal Learning in a Novel Probabilistic Reversal Learning Task for Mice
  9. Distribution of 5-HT receptors in the central nervous system: an update
  10. Synthesis and structure−activity relationships of teixobactin
  11. The BJP expects authors to share data
  12. THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: G protein-coupled receptors
  13. Metabolomics Study of the Synergistic Killing of Polymyxin B in Combination with Amikacin against Polymyxin-Susceptible and -Resistant Pseudomonas aeruginosa
  14. T-2 toxin neurotoxicity: role of oxidative stress and mitochondrial dysfunction
  15. Sex: A change in our guidelines to authors to ensure that this is no longer an ignored experimental variable
  16. The impact of backbone N ‐methylation on the structure‐activity relationship of Leu 10 ‐teixobactin
  17. Sex differences in mouse models of fear inhibition: Fear extinction, safety learning, and fear–safety discrimination
  18. Contemporary Anti-Ebola Drug Discovery Approaches and Platforms
  19. Molecular Mechanisms of Neurotoxicity Induced by Polymyxins and Chemoprevention
  20. A Comparative Study of Outer Membrane Proteome between Paired Colistin-Susceptible and Extremely Colistin-Resistant Klebsiella pneumoniae Strains
  21. Reply to Tosh et al.: Quantitative analyses of cultural evolution require engagement with historical and archaeological research
  22. Animal Models of Addiction and Neuropsychiatric Disorders and Their Role in Drug Discovery: Honoring the Legacy of Athina Markou
  23. Sputum Active Polymyxin Lipopeptides: Activity against Cystic Fibrosis Pseudomonas aeruginosa Isolates and Their Interactions with Sputum Biomolecules
  24. Experimental design and analysis and their reporting II: updated and simplified guidance for authors and peer reviewers
  25. Goals and practicalities of immunoblotting and immunohistochemistry: A guide for submission to the British Journal of Pharmacology
  26. The potentially beneficial central nervous system activity profile of ivacaftor and its metabolites
  27. Lemborexant. Dual orexin receptor antagonist, Treatment of insomnia
  28. Mechanistic Insights From Global Metabolomics Studies into Synergistic Bactericidal Effect of a Polymyxin B Combination With Tamoxifen Against Cystic Fibrosis MDR Pseudomonas aeruginosa
  29. Polymyxins for CNS infections: Pharmacology and neurotoxicity
  30. Rapamycin Confers Neuroprotection against Colistin-Induced Oxidative Stress, Mitochondria Dysfunction, and Apoptosis through the Activation of Autophagy and mTOR/Akt/CREB Signaling Pathways
  31. Orexin Receptor Antagonists
  32. THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Overview
  33. Updating the guidelines for data transparency in the British Journal of Pharmacology - data sharing and the use of scatter plots instead of bar charts
  34. 5-HT Receptor Nomenclature: Naming Names, Does It Matter? A Tribute to Maurice Rapport
  35. A short history of the 5-HT2C receptor: from the choroid plexus to depression, obesity and addiction treatment
  36. Saving, changing and repairing lives
  37. Blunted 5-HT1A receptor-mediated responses and antidepressant-like behavior in mice lacking the GABAB1a but not GABAB1b subunit isoforms
  38. Astrocytes: Adhesion Molecules and Immunomodulation
  39. Hippocampal 5-HT7receptors signal phosphorylation of the GluA1 subunit to facilitate AMPA receptor mediated-neurotransmissionin vitroandin vivo
  40. Editorial: Reporting guidelines for psychopharmacology
  41. Orexin OX2 Receptor Antagonists as Sleep Aids
  42. The Concise Guide to PHARMACOLOGY 2015/16: Overview
  43. Discovery of 1 H -pyrazolo[3,4- b ]pyridines as potent dual orexin receptor antagonists (DORAs)
  44. Experimental design and analysis and their reporting: new guidance for publication in BJP
  45. Pathological Conditions Associated with the Disturbance of the 5-HT System
  46. AQW051, a novel, potent and selective α7 nicotinic ACh receptor partial agonist: pharmacological characterization and phase I evaluation
  47. Somatostatin
  48. Suvorexant for the treatment of insomnia
  49. SOM230: A New Therapeutic Modality for Cushing's Disease
  50. Somatostatin
  51. The Concise Guide to PHARMACOLOGY 2013/14: Overview
  52. Orexin in sleep, addiction and more: Is the perfect insomnia drug at hand?
  53. An invitation for comprehensive single-compound reviews on the pharmacological properties of newly launched drugs
  54. Identification of a Novel Series of Orexin Receptor Antagonists with a Distinct Effect on Sleep Architecture for the Treatment of Insomnia
  55. Adult siRNA-induced knockdown of mGlu7 receptors reduces anxiety in the mouse
  56. Distinct effects of IPSU and suvorexant on mouse sleep architecture
  57. Kinetic properties of “dual” orexin receptor antagonists at OX1R and OX2R orexin receptors
  58. The Dual Orexin Receptor Antagonist Almorexant Induces Sleep and Decreases Orexin-Induced Locomotion by Blocking Orexin 2 Receptors
  59. Neuropeptides and Neuropeptide Receptors: Drug Targets, and Peptide and Non-Peptide Ligands: a Tribute to Prof.Dieter Seebach
  60. Neuropeptidomics of mouse hypothalamus after imipramine treatment reveal somatostatin as a potential mediator of antidepressant effects
  61. Reviewer comments on Reflections on drug research by Sir James Black
  62. Somatostatin-28 modulates prepulse inhibition of the acoustic startle response, reward processes and spontaneous locomotor activity in rats
  63. Neuropeptide receptor positive allosteric modulation in epilepsy: Galanin modulation revealed
  64. Changes of AMPA receptors in MPTP monkeys with levodopa-induced dyskinesias
  65. Decahydroisoquinoline derivatives as novel non-peptidic, potent and subtype-selective somatostatin sst3 receptor antagonists
  66. Hippocampal sst1 receptors are autoreceptors and do not affect seizures in rats
  67. Reaction of Fe3(CO)12 with octreotide—chemical, electrochemical and biological investigations
  68. Distribution of 5-HT Receptors in the Central Nervous System
  69. The mTOR kinase inhibitor Everolimus decreases S6 kinase phosphorylation but fails to reduce mutant huntingtin levels in brain and is not neuroprotective in the R6/2 mouse model of Huntington's disease
  70. NMR-Solution Structures and Affinities for the Human Somatostatin G-Protein-Coupled Receptors hsst1–5 of CF3 Derivatives of Sandostatin® (Octreotide)
  71. Somatostatin, Alzheimer's disease and cognition: An old story coming of age?
  72. Selective effects of benzodiazepines on the acquisition of conditioned taste aversion compared to attenuation of neophobia in C57BL/6 mice
  73. Novel, Potent, and Radio-Iodinatable Somatostatin Receptor 1 (sst1) Selective Analogues
  74. Discovery of novel non-peptidic β-alanine piperazine amide derivatives and their optimization to achiral, easily accessible, potent and selective somatostatin sst1 receptor antagonists
  75. New Perspective in Peptide Chemistry by N-Alkylation
  76. The selective nicotinic acetylcholine receptor α7 agonist JN403 is active in animal models of cognition, sensory gating, epilepsy and pain
  77. Increased exploratory activity of APP23 mice in a novel environment is reversed by siRNA
  78. Molecular biology of 5-HT receptors
  79. Antidepressants Influence Somatostatin Levels and Receptor Pharmacology in Brain
  80. New Open-Chain and Cyclic Tetrapeptides, Consisting ofα-,β2-, andβ3-Amino-Acid Residues, as Somatostatin Mimics - A Survey
  81. The Enantiomer of Octreotate Binds to All Five Somatostatin Receptors with Almost Equal Micromolar Affinity - A Comparison withSANDOSTATIN®
  82. Pharmacological profile of somatostatin and cortistatin receptors
  83. The Rostral Anterior Cingulate Cortex Modulates the Efficiency of Amygdala-Dependent Fear Learning
  84. Improving Oral Bioavailability of Peptides by Multiple N-Methylation: Somatostatin Analogues
  85. Ergoline derivatives as highly potent and selective antagonists at the somatostatin sst1 receptor
  86. Brain sphingosine-1-phosphate receptors: Implication for FTY720 in the treatment of multiple sclerosis
  87. mGluR7 facilitates extinction of aversive memories and controls amygdala plasticity
  88. Identification and SAR of potent and selective non-peptide obeline somatostatin sst1 receptor antagonists
  89. SAR of the arylpiperazine moiety of obeline somatostatin sst1 receptor antagonists
  90. JN403, in vitro characterization of a novel nicotinic acetylcholine receptor α7 selective agonist
  91. Emerging use of non-viral RNA interference in the brain
  92. 5-HT-5 Receptors
  93. 5-HT-6 Receptor
  94. 5-HT-7 Receptor
  95. 5-HT-1F Receptor
  96. 5-HT-3 Receptor
  97. 5-Hydroxytryptamine Receptors
  98. ABP688, a novel selective and high affinity ligand for the labeling of mGlu5 receptors: Identification, in vitro pharmacology, pharmacokinetic and biodistribution studies
  99. RNA interference as a therapeutic strategy for treating CNS disorders
  100. Region-specific transcriptional changes following the three antidepressant treatments electro convulsive therapy, sleep deprivation and fluoxetine
  101. Somatostatin receptors in wildtype and somatostatin deficient mice and their involvement in nitric oxide physiology in the retina
  102. The somatostatin sst1 receptor: an autoreceptor for somatostatin in brain and retina?
  103. Compensatory changes in the hippocampus of somatostatin knockout mice: upregulation of somatostatin receptor 2 and its function in the control of bursting activity and synaptic transmission
  104. Hyperdopaminergia and altered locomotor activity in GABAB1-deficient mice
  105. Interfering with the brain: Use of RNA interference for understanding the pathophysiology of psychiatric and neurological disorders
  106. Global Down-Regulation of Gene Expression in the Brain Using RNA Interference, with Emphasis on Monoamine Transporters and GPCRs: Implications for Target Characterization in Psychiatric and Neurological Disorders
  107. Correction: Opportunities in somatostatin research: biological, chemical and therapeutic aspects
  108. Distinct functional properties of native somatostatin receptor subtype 5 compared with subtype 2 in the regulation of ACTH release by corticotroph tumor cells
  109. siRNA-mediated knockdown of the serotonin transporter in the adult mouse brain
  110. siRNA-mediated knockdown of the serotonin transporter in the adult mouse brain
  111. Binding and functional properties of the novel somatostatin analogue KE 108 at native mouse somatostatin receptors
  112. Coupling of human nicotinic acetylcholine receptors α7 to calcium channels in GH3 cells
  113. Fish somatostatin sst3 receptor: comparison of radioligand and GTPgammaS binding, adenylate cyclase and phospholipase C activities reveals different agonist-dependent pharmacological signatures
  114. Somatostatin Receptor 1 Selective Analogues:  2. Nα-Methylated Scan†
  115. Proceedings of Neuropeptides 2004, the XIV European Neuropeptides Club meeting
  116. Neurochemical and behavioral consequences of widespread gene knockdown in the adult mouse brain by using nonviral RNA interference
  117. Somatostatin receptors differentially affect spontaneous epileptiform activity in mouse hippocampal slices
  118. Paroxetine combined with a 5-HT1A receptor antagonist reversed reward deficits observed during amphetamine withdrawal in rats
  119. The NK1 receptor antagonist NKP608 lacks anxiolytic-like activity in Swiss-Webster mice exposed to the elevated plus-maze
  120. The somatostatin receptor (sst1) modulates the release of somatostatin in the nucleus accumbens of the rat
  121. Effect of Somatostatin on Nitric Oxide Production in Human Retinal Pigment Epithelium Cell Cultures
  122. Comparison of functional profiles at human recombinant somatostatin sst2receptor: simultaneous determination of intracellular Ca2+and luciferase expression in CHO-K1 cells
  123. SRA880, in vitro characterization of the first non-peptide somatostatin sst1 receptor antagonist
  124. Applications of a Rat Multiple Tissue Gene Expression Data Set
  125. Genetic deletion of somatostatin receptor 1 alters somatostatinergic transmission in the mouse retina
  126. Withdrawal from chronic amphetamine induces Depressive-Like behavioral effects in rodents
  127. Native somatostatin sst2 and sst5 receptors functionally coupled to Gi/o-protein, but not to the serum response element in AtT-20 mouse tumour corticotrophs
  128. Pharmacological characterisation of native somatostatin receptors in AtT-20 mouse tumour corticotrophs
  129. Agonist properties of putative small-molecule somatostatin sst2 receptor-selective antagonists
  130. Biological activity of somatostatin receptors in GC rat tumour somatotrophs: evidence with sst1–sst5 receptor-selective nonpeptidyl agonists
  131. Design and Synthesis of γ-Dipeptide Derivatives with Submicromolar Affinities for Human Somatostatin Receptors
  132. β2/β3-di- and α/β3-tetrapeptide derivatives as potent agonists at somatostatin sst4 receptors
  133. Functional characterisation of the putative somatostatin sst2 receptor antagonist CYN 154806
  134. Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and hippocampal excitatory neurotransmission in mice
  135. Study of the calcium dynamics of the human α4β2, α3β4 and α1β1γδ nicotinic acetylcholine receptors
  136. Molecular, pharmacological and functional diversity of 5-HT receptors
  137. Identification and characterization of a type five-like somatostatin receptor in goldfish pituitary
  138. Somatostatin sst2 receptor knock-out mice: localisation of sst1–5 receptor mRNA and binding in mouse brain by semi-quantitative RT–PCR, in situ hybridisation histochemistry and receptor autoradiography
  139. Emerging discoveries in neuroscience: molecular bridges to the brain
  140. Pharmacological characterisation of the goldfish somatostatin sst5 receptor
  141. Drug Design at Peptide Receptors
  142. Extended Radioligand Binding Profile of Iloperidone A Broad Spectrum Dopamine/Serotonin/Norepinephrine Receptor Antagonist for the Management of Psychotic Disorders
  143. Linear, Peptidase-Resistantβ2/β3-Di- andα/β3-Tetrapeptide Derivatives with Nanomolar Affinities to a Human Somatostatin Receptor, Preliminary Communication
  144. Lack of evidence for cross-competition between vasoactive intestinal peptide and somatostatin at their respective receptors
  145. Peptide Folding Induces High and Selective Affinity of a Linear and Small β-Peptide to the Human Somatostatin Receptor 4
  146. Distribution and characterisation of somatostatin receptor mRNA and binding sites in the brain and periphery
  147. Recovery of emotional behaviour in neural cell adhesion molecule (NCAM) null mutant mice through transgenic expression of NCAM180
  148. Cloning, expression and pharmacological characterisation of the mouse somatostatin sst5 receptor
  149. Syntheses and biological activities of sandostatin analogs containing stereochemical changes in positions 6 or 8
  150. Cloning, expression, functional coupling and pharmacological characterization of the rat dopamine D 4 receptor
  151. Potent and Selective Non-Peptidic Inhibitors of Endothelin-Converting Enzyme-1 with Sustained Duration of Action
  152. The Cyclo-β-Tetrapeptide (β-HPhe-β-HThr-β-HLys-β-HTrp): Synthesis, NMR Structure in Methanol Solution, and Affinity for Human Somatostatin Receptors
  153. Characterisation of human recombinant somatostatin receptors. 1. Radioligand binding studies
  154. Characterisation of human recombinant somatostatin receptors. 2. Modulation of GTPγS binding
  155. Characterisation of human recombinant somatostatin receptors. 3. Modulation of adenylate cyclase activity
  156. Characterisation of human recombinant somatostatin receptors. 4. Modulation of phospholipase C activity
  157. Brain somatostatin: a candidate inhibitory role in seizures and epileptogenesis
  158. Receptor density as a factor governing the efficacy of the dopamine D4receptor ligands, L-745,870 and U-101958 at human recombinant D4.4receptors expressed in CHO cells
  159. Anxiety and increased 5-HT1A receptor response in NCAM null mutant mice
  160. Molecular Cloning and Pharmacological Characterization of a Somatostatin Receptor Subtype in the Gymnotiform Fish Apteronotus albifrons
  161. Pharmacological characterisation of 5-HT receptors positively coupled to adenylyl cyclase in the rat hippocampus
  162. Structural and compositional determinants of cortistatin activity
  163. Synthesis and Biological Evaluation of a Cyclo--tetrapeptide as a Somatostatin Analogue
  164. Characterisation of the fish sst3 receptor, a member of the SRIF1 receptor family: atypical pharmacological features
  165. Preface
  166. High Affinity of SDZ HTF-919 and Related Molecules for Calf and Human Caudate 5-HT4 Receptors
  167. Impact of the Human Genome Project on the Principles for Classification and Nomenclature of 5-HT Receptors
  168. The role ofα2-adrenoceptor antagonism in the anti-cataleptic properties of the atypical neuroleptic agent, clozapine, in the rat
  169. Design, Synthesis, and Biological Activities of Potent and Selective Somatostatin Analogues Incorporating Novel Peptoid Residues
  170. The agonist activities of the putative antipsychotic agents, L-745,870 and U-101958 in HEK293 cells expressing the human dopamine D4.4receptor
  171. [125I]Tyr10-cortistatin14 labels all five somatostatin receptors
  172. [][Tyr3]octreotide labels human somatostatin sst2 and sst5 receptors
  173. The structure and signalling properties of 5-HT receptors: an endless diversity?
  174. Identification and pharmacological characterization of somatostatin receptors in rat lung
  175. 5-HT Receptor Classification and Nomenclature: Towards a Harmonization with the Human Genome
  176. Editorial
  177. Inhibition of cAMP Accumulation Via Recombinant Human Serotonin 5-HT 1A Receptors: Considerations on Receptor Effector Coupling across Systems
  178. Autoradiographic analysis of somatostatin SRIF1 and SRIF2 receptors in the human brain and pituitary
  179. Pharmacological characterisation of human cerebral cortex somatostatin SRIF1 and SRIF2 receptors
  180. Minireview: Nomenclature and Classification of Transmitter Receptors: an Integrated Approach
  181. Presence of somatostatin sst2 receptors in the developing rat auditory system
  182. Status of somatostatin receptor messenger RNAs and binding sites in rat brain during kindling epileptogenesis
  183. Binding properties of somatostatin receptor subtypes
  184. Somatostatin receptors in the Rhesus monkey brain: localization and pharmacological characterization
  185. Alignment of receptor nomenclature with the human genome: classification of 5-HT1B and 5-HT1D receptor subtypes
  186. Somatostatin receptors in the developing rat brain
  187. Classification and nomenclature of 5-HT receptors: a comment on current issues
  188. Embryonic and postnatal mRNA distribution of five somatostatin receptor subtypes in the rat brain
  189. Localization of the 5-hydroxytryptamine2C receptor protein in human and rat brain using specific antisera
  190. The Serotonin 5-HT4 Receptor. 1. Design of a New Class of Agonists and Receptor Map of the Agonist Recognition Site
  191. The Serotonin 5-HT4 Receptor. 2. Structure-Activity Studies of the Indole Carbazimidamide Class of Agonists
  192. Functional effects of d-Phe-c[Cys-Tyr-d-Trp-Lys-Val-Cys]-Trp-NH2 and differential changes in somatostatin receptor messenger RNAs, binding sites and somatostatin release in kainic acid-treated rats
  193. Characterization and distribution of somatostatin SS-1 and SRIF-1 binding sites in rat brain: identitity with SSTR-2 receptors
  194. Classification and nomenclature of somatostatin receptors
  195. Pharmacological identity between somatostatin SS-2 binding sites and SSTR-1 receptors
  196. Co-expression of somatostatin SSTR-3 and SSTR-4 receptor messenger RNAs in the rat brain
  197. Molecular pharmacology of somatostatin receptors
  198. Chromic mianserin or eltoprazine treatment in rats: effects on the elevated plus-maze test and on limbic 5-HT2C receptor levels
  199. Molecular Pharmacology of Somatostatin-receptor Subtypes
  200. Localization of 5-HT1B, 5-HT1Dα, 5-HT1E and 5-HT1F receptor messenger RNA in rodent and primate brain
  201. Localization of somatostatin (SRIF) SSTR-1, SSTR-2 and SSTR-3 receptor mRNA in rat brain by in situ hybridization
  202. A comparative autoradiographic study of 5-HT1D binding sites in human and guinea-pig brain using different radioligands
  203. Effect of 5,7-dihydroxytryptamine lesion on mianserin-induced conditioned place aversion and on 5-hydroxytryptamine1C receptors in the rat brain
  204. Endothelin receptors in the human coronary artery, ventricle and atrium
  205. Distribution and second messenger coupling of four somatostatin receptor subtypes expressed in brain
  206. Calcineurin inhibits desensitization of cloned rat 5-HT1C receptors
  207. Partial agonists, full agonists, antagonists: dilemmas of definition
  208. The novel 5-HT1A receptor antagonist, SDZ 216-525, decreases 5-HT release in rat hippocampus in vivo
  209. A proposed new nomenclature for 5-HT receptors
  210. Autoradiographic characterisation and localisation of 5-HT1D compared to 5-HT1B binding sites in rat brain
  211. 5-Hydroxytryptamine1 recognition sites in rat brain: Heterogeneity of non-5-hydroxytryptamine1a/1c binding sites revealed by quantitative receptor autoradiography
  212. SDZ 216–525, a selective and potent 5-HT1A receptor antagonist
  213. Evidence for the presence of 5-HT1B receptor messenger RNA in neurons of the rat trigeminal ganglia
  214. Agonist/antagonist interactions with cloned human 5-HT1A receptors: variations in intrinsic activity studied in transfected HeLa cells
  215. Direct visualization of serotonin1D receptors in the human brain using a new iodinated radioligand
  216. 5-Hydroxytryptamine (5-HT) receptor superfamilies
  217. Homogeneous 5-HT1D recognition sites in the human substantia nigra identified with a new iodinated radioligand
  218. Competitive antagonism by recognised 5-HT2 receptor antagonists at 5-HT1C receptors in pig choroid plexus
  219. Interaction of the α-adrenoceptor agonist oxymetazoline with serotonin 5-HT1A, 5-HT1B, 5-HT1C and 5-HT1D receptors
  220. 5-HT1-like receptors mediate 5-hydroxytryptamine-induced contraction of guinea-pig isolated iliac artery
  221. Receptor biochemistry and methodology volume 15: Serotonin receptor subtypes
  222. 5-HT Receptors: Subtypes and Second Messengers
  223. Autoradiography of 5-HT receptors: A critical appraisal
  224. Distribution of Serotonin Receptors
  225. The serotonin 5-HT1D receptor: A progress review
  226. Receptor modification in the brains of spontaneously hypertensive and Wistar-Kyoto rats: regionally specific and selective increase in cerebellar beta 2-adrenoceptors.
  227. Similar distribution of [125I]sarafotoxin-6b and [125I]endothelin-1, -2, -3 binding sites in the human kidney
  228. Selective Agonists and Antagonists at 5-Hydroxytryptamine Receptor Subtypes
  229. Subtypes of α1-adrenoceptors in hippocampus of pigs, guinea-pigs, calves and humans: regional differences
  230. Interaction of psychotropic drugs with central 5-HT3 recognition sites: fact or artifact?
  231. Is the sumatripan (GR 43175)-induced endothelium-dependent relaxation of pig coronary arteries mediated by 5-HT1D receptors?
  232. The pharmacological properties of the presynaptic serotonin autoreceptor in the pig brain cortex conform to the 5-HT1D receptor subtype
  233. Species differences in the pharmacology of terminal 5-HT autoreceptors in mammalian brain
  234. 5-Hydroxytryptamine3 receptors in the human brain: Autoradiographic visualization using [3H]ICS 205-930
  235. Competitive Interaction of Agonists and Antagonists with 5-HT3-Recognition Sites in Membranes of Neuroblastoma Cells Labelled with [3H] ICS 205–930
  236. Localisation by autoradiography of neuronal 5-HT3 receptors in the mouse CNS
  237. Molecular pharmacology of 5-HT1D recognition sites: Radioligand binding studies in human, pig and calf brain membranes
  238. The 5-hydroxytryptamine 5-HT1D receptor subtype is negatively coupled to adenylate cyclase in calf substantia nigra
  239. Characterisation of 5-HT3 recognition sites in membranes of NG 108-15 neuroblastoma-glioma cells with [3H]ICS 205-930
  240. Visualization of a novel serotonin recognition site (5-HT1D) in the human brain by autoradiography
  241. [125I]SCH 23982, a ‘selective’ D-1 receptor antagonist, labels with high affinity 5-HT1C sites in pig choroid plexus
  242. Central 5-HT1A Receptors and the Mechanism of the Central Hypotensive Effect of (+)8-OH-DPAT, DP-5-CT, R28935, and Urapidil
  243. Identification of a 5-HT1 recognition site in human brain membranes different from 5-HT1A, 5-HT1B and 5-HT1C sites
  244. Molecular pharmacology and biology of 5-HT1C receptors
  245. 5-HT1D receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in calf substantia nigra
  246. Functional Correlates of Serotonin 5-HT1Recognition Sites
  247. Identification of serotonin 5-HT3 recognition sites by radioligand binding in NG108-15 neuroblastoma-glioma cells
  248. α1-adrenoceptors in the mammalian brain: similar pharmacology but different distribution in rodents and primates
  249. [3H]Ketanserin labels 5-HT2 receptors and ?1-adrenoceptors in human and pig brain membranes
  250. Inhibition of 5-carboxamidotryptamine-induced relaxation of guinea-pig ileum correlates with [125I]LSD binding
  251. 5-HT1A-receptors mediate stimulation of adenylate cyclase in rat hippocampus
  252. Serotonin increases the production of inositol phosphates and mobilises calcium via the 5-HT2 receptor in A7r5 smooth muscle cells
  253. Serotonin receptors in the human brain. I. Characterization and autoradiographic localization of 5-HT1A recognition sites. Apparent absence of 5-HT1B recognition sites
  254. Serotonin receptors in the human brain. II. Characterization and autoradiographic localization of 5-HT1C and 5-HT2 recognition sites
  255. Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites
  256. Implications of stereoselectivity in radioligand binding studies
  257. Characterization of the 5-HTIB recognition site in rat brain: Binding studies with (−)[125I]Iodocyanopindolol
  258. Molecular pharmacology of 5-HT1 and 5-HT2 recognition sites in rat and pig brain membranes: Radioligand binding studies with [3H]5-HT, [3H]8-OH-DPAT, (−)[125I]iodocyanopindolol, [3H]mesulergine and [3H]Ketanserin
  259. Mesulergine, a selective serotonin-2 ligand in the rat cortex, does not label these receptors in porcine and human cortex: Evidence for species differences in brain serotonin-2 receptors
  260. The binding of serotonergic ligands to the porcine choroid plexus: Characterization of a new type of serotonin recognition site
  261. Characterization of IBE 2254 Binding to Alpha - Adrenergic Receptors on Intact DDT Smooth Muscle Cells: Comparison with Membrane1Binding and Correlation with Phosphoinositides Breakdown
  262. Identification of 5HT2-Receptors on Longitudinal Muscle of the Guinea Pig Ileum
  263. Binding of125I-Cyanopindolol to Beta-1-Adreno-Ceptors in a High and Low Affinity State
  264. Non-specific uptake of the radioligand 125I-IHYP by intact human lymphocytes: Reversal of the uptake process
  265. Binding characteristics of (+)-, (�)- and (-)-[125Iodo] cyanopindolol to guinea-pig left ventricle membranes
  266. (�)[125Iodo]cyanopindolol, a new ligand for ?-adrenoceptors: Identification and quantitation of subclasses of ?-adrenoceptors in guinea pig
  267. The β-adrenergic receptor in human lymphocytes: Subclassification by the use of a new radio-ligand, (±)−125iodocyanopindolol
  268. [125I]BE 2254, a new high affinity radioligand for α1-adrenoceptors
  269. Assessing allosteric ligand-receptor interactions
  270. Molecular biology of 5-HT receptors
  271. Highly N-Methylated Somatostatin Analogs: Synthesis, Biological Activity and Structure-Activity Relationship Studies
  272. Serotoninergic System
  273. Somatostatin Receptor Gene Family - Subtype Selectivity for Ligand Binding