All Stories

  1. Regioselective Synthesis of Potential Non-Quinonoid Prodrugs of Plasmodione: Antiparasitic Properties Against Two Hemoglobin-Feeding Parasites and Drug Metabolism Studies

    Article • Molecules, November 2024, MDPI AG

    Elisabeth Davioud-Charvet

  2. Chemoselective Synthesis and Anti-Kinetoplastidal Properties of 2,6-Diaryl-4H-tetrahydro-thiopyran-4-one S-Oxides: Their Interplay in a Cascade of Redox Reactions from Diarylideneacetones

    Article • Molecules, April 2024, MDPI AG

    Elisabeth Davioud-Charvet

  3. Synthesis and Photochemical Properties of Fluorescent Metabolites Generated from Fluorinated Benzoylmenadiones in Living Cells

    Article • The Journal of Organic Chemistry, June 2023, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  4. Evaluation of ferrocenyl-containing γ-hydroxy-γ-lactam-derived tetramates as potential antiplasmodials

    Article • European Journal of Medicinal Chemistry, December 2022, Elsevier

    Elisabeth Davioud-Charvet

  5. Efficient Multigram-Scale Synthesis of 7-Substituted 3-Methyltetral-1-ones and 6-Fluoromenadione

    Article • Organic Process Research & Development, February 2022, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  6. The parasitophorous vacuole nutrient channel is critical for drug access in malaria parasites and modulates the artemisinin resistance fitness cost

    Article • Cell Host & Microbe, December 2021, Elsevier

    Elisabeth Davioud-Charvet

  7. Bioinspired Photoredox Benzylation of Quinones

    Article • The Journal of Organic Chemistry, July 2021, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  8. Direct C−H Radical Alkylation of 1,4‐Quinones

    Article • European Journal of Organic Chemistry, July 2021, Wiley

    Elisabeth Davioud-Charvet

  9. Magnesium Complexes of Ladanein: A Beneficial Strategy for Stabilizing Polyphenolic Antivirals

    Article • European Journal of Inorganic Chemistry, July 2021, Wiley

    Elisabeth Davioud-Charvet

  10. A Class of Valuable (Pro-)Activity-Based Protein Profiling Probes: Application to the Redox-Active Antiplasmodial Agent, Plasmodione

    Article • JACS Au, April 2021, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  11. Plasmodium falciparum Ferredoxin-NADP+ Reductase-Catalyzed Redox Cycling of Plasmodione Generates Both Predicted Key Drug Metabolites: Implication for Antimalarial Drug Development

    Article • ACS Infectious Diseases, April 2021, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  12. Repurposing Auranofin and Evaluation of a New Gold(I) Compound for the Search of Treatment of Human and Cattle Parasitic Diseases: From Protozoa to Helminth Infections

    Article • Molecules, November 2020, MDPI AG

    Elisabeth Davioud-Charvet

  13. A role for the succinate dehydrogenase in the mode of action of the redox-active antimalarial drug, plasmodione

    Article • Free Radical Biology and Medicine, November 2020, Elsevier

    Elisabeth Davioud-Charvet

  14. A Mild and Versatile Friedel–Crafts Methodology for the Diversity‐Oriented Synthesis of Redox‐Active 3‐Benzoylmenadiones with Tuneable Redox Potentials

    Article • Chemistry - A European Journal, January 2020, Wiley

    Elisabeth Davioud-Charvet

  15. A Mild and Versatile Friedel–Crafts Methodology for the Diversity‐Oriented Synthesis of Redox‐Active 3‐Benzoylmenadiones with Tunable Redox Potentials

    Article • Chemistry - A European Journal, January 2020, Wiley

    Elisabeth Davioud-Charvet

  16. Antiplasmodial Activity of Nitroaromatic Compounds: Correlation with Their Reduction Potential and Inhibitory Action on Plasmodium falciparum Glutathione Reductase

    Article • Molecules, December 2019, MDPI AG

    Elisabeth Davioud-Charvet

  17. Investigating the mode of action of the redox-active antimalarial drug plasmodione using the yeast model

    Article • Free Radical Biology and Medicine, September 2019, Elsevier

    Elisabeth Davioud-Charvet

  18. Selenium Status in Elderly People: Longevity and Age-Related Diseases

    Article • Current Pharmaceutical Design, August 2019, Bentham Science Publishers

    Elisabeth Davioud-Charvet

  19. Author Correction: Arylmethylamino steroids as antiparasitic agents

    Article • Nature Communications, July 2019, Springer Science + Business Media

    Elisabeth Davioud-Charvet

  20. Physicochemical Properties Govern the Activity of Potent Antiviral Flavones

    Article • ACS Omega, March 2019, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  21. AntiMalarial Mode of Action (AMMA) Database: Data Selection, Verification and Chemical Space Analysis

    Article • Molecular Informatics, May 2018, Wiley

    Elisabeth Davioud-Charvet

  22. Synthesis of plasmodione metabolites and13C-enriched plasmodione as chemical tools for drug metabolism investigation

    Article • Organic & Biomolecular Chemistry, January 2018, Royal Society of Chemistry

    Elisabeth Davioud-Charvet

  23. Iron(iii) coordination properties of ladanein, a flavone lead with a broad-spectrum antiviral activity

    Article • New Journal of Chemistry, January 2018, Royal Society of Chemistry

    Elisabeth Davioud-Charvet

  24. QSAR modeling and chemical space analysis of antimalarial compounds

    Article • Journal of Computer-Aided Molecular Design, April 2017, Springer Science + Business Media

    Elisabeth Davioud-Charvet

  25. A high susceptibility to redox imbalance of the transmissible stages of Plasmodium falciparum revealed with a luciferase‐based mature gametocyte assay

    Article • Molecular Microbiology, February 2017, Wiley

    Elisabeth Davioud-Charvet, Professor David A Fidock

  26. Arylmethylamino steroids as antiparasitic agents

    Article • Nature Communications, February 2017, Nature

    Elisabeth Davioud-Charvet

  27. Pharmacomodulation of the Antimalarial Plasmodione: Synthesis of Biaryl- and N-Arylalkylamine Analogues, Antimalarial Activities and Physicochemical Properties

    Article • Molecules, January 2017, MDPI AG

    Elisabeth Davioud-Charvet

  28. A Redox-Active Fluorescent pH Indicator for Detecting Plasmodium falciparum Strains with Reduced Responsiveness to Quinoline Antimalarial Drugs

    Article • ACS Infectious Diseases, December 2016, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  29. ChemInform Abstract: A Platform of Regioselective Methodologies to Access Polysubstituted 2-Methyl-1,4-naphthoquinone Derivatives: Scope and Limitations.

    Article • ChemInform, August 2016, Wiley

    Elisabeth Davioud-Charvet

  30. In Silico Mining for Antimalarial Structure-Activity Knowledge and Discovery of Novel Antimalarial Curcuminoids

    Article • Molecules, June 2016, MDPI AG

    Elisabeth Davioud-Charvet

  31. The Redox Cycler Plasmodione Is a Fast-Acting Antimalarial Lead Compound with Pronounced Activity against Sexual and Early Asexual Blood-Stage Parasites

    Article • Antimicrobial Agents and Chemotherapy, June 2016, ASM Journals

    Elisabeth Davioud-Charvet

  32. A Platform of Regioselective Methodologies to Access Polysubstituted 2-Methyl-1,4-naphthoquinone Derivatives: Scope and Limitations

    Article • European Journal of Organic Chemistry, March 2016, Wiley

    Elisabeth Davioud-Charvet

  33. Redox Polypharmacology as an Emerging Strategy to Combat Malarial Parasites

    Article • ChemMedChem, March 2016, Wiley

    Elisabeth Davioud-Charvet

  34. Synthesis and evaluation of 1,4-naphthoquinone ether derivatives asSmTGR inhibitors and new anti-schistosomal drugs

    Article • FEBS Journal, August 2015, Wiley

    Elisabeth Davioud-Charvet

  35. ChemInform Abstract: Diastereoselective Synthesis of 2,6-Diaryltetrahydrothiopyran-4-ones by Phase-Transfer Catalysis.

    Article • ChemInform, June 2015, Wiley

    Elisabeth Davioud-Charvet

  36. Antimalarial NADPH-Consuming Redox-Cyclers As Superior Glucose-6-Phosphate Dehydrogenase Deficiency Copycats

    Article • Antioxidants & Redox Signaling, May 2015, Mary Ann Liebert Inc

    Elisabeth Davioud-Charvet

  37. Diastereoselective Synthesis of 2,6-Diaryltetrahydrothiopyran-4-ones by Phase-Transfer Catalysis

    Article • European Journal of Organic Chemistry, February 2015, Wiley

    Elisabeth Davioud-Charvet

  38. Electrochemical Properties of Substituted 2-Methyl-1,4-Naphthoquinones: Redox Behavior Predictions

    Article • Chemistry - A European Journal, December 2014, Wiley

    Elisabeth Davioud-Charvet

  39. Antiglioma activity of GoPI-sugar, a novel gold(I)–phosphole inhibitor: Chemical synthesis, mechanistic studies, and effectiveness in vivo

    Article • Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics, August 2014, Elsevier

    Elisabeth Davioud-Charvet

  40. A Practical and Economical High-Yielding, Six-Step Sequence Synthesis of a Flavone: Application to the Multigram-Scale Synthesis of Ladanein

    Article • Organic Process Research & Development, May 2014, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  41. Versatile Synthesis of Dissymmetric Diarylideneacetones via a Palladium-Catalyzed­ Coupling-Isomerization Reaction

    Article • Synthesis, April 2013, Thieme Publishing Group

    Elisabeth Davioud-Charvet, Professor Thomas J J Müller

  42. ChemInform Abstract: Versatile Synthesis of Dissymmetric Diarylideneacetones via a Palladium-Catalyzed Coupling-Isomerization Reaction.

    Article • ChemInform, April 2013, Wiley

    Elisabeth Davioud-Charvet

  43. Redox-Active Agents in Reactions Involving the Trypanothione/Trypanothione Reductase-based System to Fight Kinetoplastidal Parasites

    Article • April 2013, Wiley

    Elisabeth Davioud-Charvet

  44. 1,4-Naphthoquinones and Other NADPH-Dependent Glutathione Reductase- Catalyzed Redox Cyclers as Antimalarial Agents

    Article • Current Pharmaceutical Design, March 2013, Bentham Science Publishers

    Elisabeth Davioud-Charvet

  45. The Antimalarial Activities of Methylene Blue and the 1,4-Naphthoquinone 3-[4-(Trifluoromethyl)Benzyl]-Menadione Are Not Due to Inhibition of the Mitochondrial Electron Transport Chain

    Article • Antimicrobial Agents and Chemotherapy, February 2013, ASM Journals

    Elisabeth Davioud-Charvet

  46. Drug Discovery in Infectious Diseases, Volume 3: Parasitic Helminths: Targets, Screens, Drugs and Vaccines. Edited by Conor R. Caffrey

    Article • ChemMedChem, November 2012, Wiley

    Elisabeth Davioud-Charvet

  47. Versatile Synthesis of Dissymmetric Diarylideneacetones via a Palladium-Catalyzed­ Coupling–Isomerization Reaction

    Article • Synthesis, November 2012, Thieme Publishing Group

    Elisabeth Davioud-Charvet, Professor Thomas J J Müller

  48. Interactions of the Antimalarial Drug Methylene Blue with Methemoglobin and Heme Targets inPlasmodium falciparum: A Physico-Biochemical Study

    Article • Antioxidants & Redox Signaling, August 2012, Mary Ann Liebert Inc

    Elisabeth Davioud-Charvet

  49. A Plant-Derived Flavonoid Inhibits Entry of All HCV Genotypes Into Human Hepatocytes

    Article • Gastroenterology, July 2012, Elsevier

    Elisabeth Davioud-Charvet, Ralf Bartenschlager

  50. Synthesis and biological evaluation of 1,4-naphthoquinones and quinoline-5,8-diones as antimalarial and schistosomicidal agents

    Article • Organic & Biomolecular Chemistry, January 2012, Royal Society of Chemistry

    Elisabeth Davioud-Charvet

  51. Exploring the trifluoromenadione core as a template to design antimalarial redox-active agents interacting with glutathione reductase

    Article • Organic & Biomolecular Chemistry, January 2012, Royal Society of Chemistry

    Elisabeth Davioud-Charvet

  52. Glutathione Reductase-Catalyzed Cascade of Redox Reactions To Bioactivate Potent Antimalarial 1,4-Naphthoquinones – A New Strategy to Combat Malarial Parasites

    Article • Journal of the American Chemical Society, August 2011, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  53. Subversive Substrates of Glutathione Reductases from Plasmodium falciparum-Infected Red Blood Cells as Antimalarial Agents

    Article • February 2011, Wiley

    Elisabeth Davioud-Charvet

  54. ChemInform Abstract: New Steroidal Diazo Ketones as Potential Photoaffinity Labeling Reagents for the Mineralocorticoid Receptor: Synthesis and Biological Activities.

    Article • ChemInform, August 2010, Wiley

    Elisabeth Davioud-Charvet

  55. ChemInform Abstract: New Potent Inhibitors of Trypanothione Reductase from Trypanosoma cruzi in the 2-Aminodiphenylsulfide Series.

    Article • ChemInform, August 2010, Wiley

    Elisabeth Davioud-Charvet

  56. ChemInform Abstract: Structure-Activity Relationships in 2-Aminodiphenylsulfides Against Trypanothione Reductase from Trypanosoma cruzi.

    Article • ChemInform, June 2010, Wiley

    Elisabeth Davioud-Charvet

  57. ChemInform Abstract: A General Approach to the Synthesis of Polyamine Linked-Monoindolylmaleimides, a New Series of Trypanothione Reductase Inhibitors.

    Article • ChemInform, June 2010, Wiley

    Elisabeth Davioud-Charvet

  58. ChemInform Abstract: Automated Parallel Synthesis of a Tetrahydroisoquinolin-Based Library: Potential Prolyl Endopeptidase Inhibitors.

    Article • ChemInform, June 2010, Wiley

    Elisabeth Davioud-Charvet

  59. Antimalarial versus Cytotoxic Properties of Dual Drugs Derived From 4-Aminoquinolines and Mannich Bases: Interaction with DNA

    Article • Journal of Medicinal Chemistry, April 2010, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  60. 752 INHIBITION OF HEPATITS C VIRUS ENTRY BY A PLANT-DERIVED FLAVONE

    Article • Journal of Hepatology, April 2010, Elsevier

    Elisabeth Davioud-Charvet

  61. Antimalarial activities of ferroquine conjugates with either glutathione reductase inhibitors or glutathione depletors via a hydrolyzable amide linker

    Article • Bioorganic & Medicinal Chemistry, December 2009, Elsevier

    Elisabeth Davioud-Charvet

  62. Unsaturated Mannich Bases Active Against Multidrug-ResistantTrypanosoma brucei bruceiStrains

    Article • ChemMedChem, March 2009, Wiley

    Elisabeth Davioud-Charvet, Professor Thomas J J Müller

  63. A Sugar-Modified Phosphole Gold Complex with Antiproliferative Properties Acting as a Thioredoxin Reductase Inhibitor in MCF-7 Cells

    Article • ChemMedChem, November 2008, Wiley

    Elisabeth Davioud-Charvet

  64. Antimalarial Dual Drugs Based on Potent Inhibitors of Glutathione Reductase fromPlasmodium falciparum

    Article • Journal of Medicinal Chemistry, March 2008, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  65. The aza-analogues of 1,4-naphthoquinones are potent substrates and inhibitors of plasmodial thioredoxin and glutathione reductases and of human erythrocyte glutathione reductase

    Article • Organic & Biomolecular Chemistry, January 2008, Royal Society of Chemistry

    Elisabeth Davioud-Charvet

  66. Correction: Thioredoxin Glutathione Reductase from Schistosoma mansoni: An Essential Parasite Enzyme and a Key Drug Target

    Article • PLoS Medicine, August 2007, PLOS

    Elisabeth Davioud-Charvet, Elias Arner

  67. Thioredoxin Glutathione Reductase from Schistosoma mansoni: An Essential Parasite Enzyme and a Key Drug Target

    Article • PLoS Medicine, June 2007, PLOS

    Elisabeth Davioud-Charvet, Elias Arner

  68. Crystal Structure of human Glutathione Reductase complexed with a Fluoro-Analogue of the Menadione Derivative M5

    Article • September 2006, Protein Data Bank, Rutgers University

    Elisabeth Davioud-Charvet

  69. A Fluoro Analogue of the Menadione Derivative 6-[2‘-(3‘-Methyl)-1‘,4‘-naphthoquinolyl]hexanoic Acid Is a Suicide Substrate of Glutathione Reductase. Crystal Structure of the Alkylated Human Enzyme†

    Article • Journal of the American Chemical Society, August 2006, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  70. Specific Inhibitors of Plasmodium falciparum Thioredoxin Reductase as Potential Antimalarial Agents.

    Article • ChemInform, July 2006, Wiley

    Elisabeth Davioud-Charvet

  71. Crystal Structure Analysis of the human Glutahione Reductase, complexed with GoPI

    Article • April 2006, Protein Data Bank, Rutgers University

    Elisabeth Davioud-Charvet

  72. Specific inhibitors of Plasmodium falciparum thioredoxin reductase as potential antimalarial agents

    Article • Bioorganic & Medicinal Chemistry Letters, April 2006, Elsevier

    Elisabeth Davioud-Charvet

  73. Gold(I)-Phosphinkomplexe für die irreversible Hemmung von humanen Disulfid-Reduktasen

    Article • Angewandte Chemie International Edition, March 2006, Wiley

    Elisabeth Davioud-Charvet

  74. Undressing of Phosphine Gold(I) Complexes as Irreversible Inhibitors of Human Disulfide Reductases

    Article • Angewandte Chemie International Edition, March 2006, Wiley

    Elisabeth Davioud-Charvet

  75. Irreversible Inactivation of Trypanothione Reductase by Unsaturated Mannich Bases:  A Divinyl Ketone as Key Intermediate

    Article • Journal of Medicinal Chemistry, November 2005, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  76. Synthesis of 5-Nitro-2-furancarbohydrazides and Theircis-Diamminedichloroplatinum Complexes as Bitopic and Irreversible Human Thioredoxin Reductase Inhibitors

    Article • Journal of Medicinal Chemistry, November 2005, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  77. Mechanistic Studies on a Novel, Highly Potent Gold-Phosphole Inhibitor of Human Glutathione Reductase

    Article • Journal of Biological Chemistry, March 2005, American Society for Biochemistry & Molecular Biology (ASBMB)

    Elisabeth Davioud-Charvet

  78. 5-Substituted Tetrazoles as Bioisosteres of Carboxylic Acids. Bioisosterism and Mechanistic Studies on Glutathione Reductase Inhibitors as Antimalarials

    Article • Journal of Medicinal Chemistry, November 2004, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  79. Screening of Plasmodium falciparum iron superoxide dismutase inhibitors and accuracy of the SOD-assays

    Article • Bioorganic & Medicinal Chemistry, November 2003, Elsevier

    Elisabeth Davioud-Charvet

  80. Mechanism-Based Inactivation of Thioredoxin Reductase fromPlasmodium falciparumby Mannich Bases. Implication for Cytotoxicity†

    Article • Biochemistry, November 2003, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  81. Double-drug development against antioxidant enzymes fromPlasmodium falciparum

    Article • Redox Report, October 2003, Taylor & Francis

    Elisabeth Davioud-Charvet

  82. Antitrypanosomal Activities and Cytotoxicity of 5-Nitro-2-furancarbohydrazides.

    Article • ChemInform, April 2003, Wiley

    Elisabeth Davioud-Charvet

  83. A novel mechanism for inhibition of HIV-1 reverse transcriptase

    Article • Bioorganic Chemistry, December 2002, Elsevier

    Elisabeth Davioud-Charvet

  84. Antitrypanosomal activities and cytotoxicity of 5-nitro-2-furancarbohydrazides

    Article • Bioorganic & Medicinal Chemistry Letters, December 2002, Elsevier

    Elisabeth Davioud-Charvet

  85. Comparison of the Inhibition of Human and Trypanosoma cruzi Prolyl Endopeptidases

    Article • Bioorganic & Medicinal Chemistry, June 2002, Elsevier

    Elisabeth Davioud-Charvet

  86. A Prodrug Form of aPlasmodium falciparumGlutathione Reductase Inhibitor Conjugated with a 4-Anilinoquinoline

    Article • Journal of Medicinal Chemistry, November 2001, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  87. Trypanosoma cruzi Prolyl Oligopeptidase Tc80 Is Involved in Nonphagocytic Mammalian Cell Invasion by Trypomastigotes

    Article • Journal of Biological Chemistry, October 2001, American Society for Biochemistry & Molecular Biology (ASBMB)

    Elisabeth Davioud-Charvet

  88. Bromination Studies of the 2,3-Dimethylnaphthazarin Core Allowing Easy Access to Naphthazarin Derivatives

    Article • The Journal of Organic Chemistry, August 2001, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  89. Antiplasmodial Activity and Cytotoxicity of Bis-, Tris-, and Tetraquinolines with Linear or Cyclic Amino Linkers

    Article • Journal of Medicinal Chemistry, May 2001, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  90. Potent and specific inhibitors of trypanothione reductase from Trypanosoma cruzi

    Article • Bioorganic & Medicinal Chemistry, April 2001, Elsevier

    Elisabeth Davioud-Charvet

  91. 2- and 3-Substituted 1,4-Naphthoquinone Derivatives as Subversive Substrates of Trypanothione Reductase and Lipoamide Dehydrogenase fromTrypanosomacruzi:  Synthesis and Correlation between Redox Cycling Activities and in Vitro Cytotoxicity

    Article • Journal of Medicinal Chemistry, February 2001, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  92. The conserved redox-sensitive cysteine residue of the DNA-binding region in the c-Rel protein is involved in the regulation of the phosphorylation of the protein

    Article • Biochemical Journal, December 2000, Portland Press Ltd.

    Elisabeth Davioud-Charvet

  93. The conserved redox-sensitive cysteine residue of the DNA-binding region in the c-Rel protein is involved in the regulation of the phosphorylation of the protein

    Article • Biochemical Journal, December 2000, Portland Press Ltd.

    Elisabeth Davioud-Charvet

  94. Antimalarial, Antitrypanosomal, and Antileishmanial Activities and Cytotoxicity of Bis(9-amino-6-chloro-2-methoxyacridines):  Influence of the Linker#

    Article • Journal of Medicinal Chemistry, July 2000, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  95. Parallel synthesis of a library of 1,4-naphthoquinones and automated screening of potential inhibitors of trypanothione reductase from Trypanosoma cruzi

    Article • Bioorganic & Medicinal Chemistry Letters, April 2000, Elsevier

    Elisabeth Davioud-Charvet

  96. Trypanothione reductase inhibition/trypanocidal activity relationships in a 1,4-bis(3-aminopropyl)piperazine series

    Article • Bioorganic & Medicinal Chemistry, January 2000, Elsevier

    Elisabeth Davioud-Charvet

  97. Synthesis of polyamine derivatives for the preparation of affinity chromatography columns for the search of new Trypanosoma cruzi targets

    Article • Bioorganic & Medicinal Chemistry Letters, June 1999, Elsevier

    Elisabeth Davioud-Charvet

  98. Synthesis of 5,5′-Dithiobis(2-nitrobenzamides)as Alternative Substrates for Trypanothione Reductase and Thioredoxin Reductase: A Microtiter Colorimetric Assay for Inhibitor Screening

    Article • Analytical Biochemistry, March 1999, Elsevier

    Elisabeth Davioud-Charvet

  99. Automated parallel synthesis of a tetrahydroisoquinolin-based library: Potential prolyl endopeptidase inhibitors

    Article • Bioorganic & Medicinal Chemistry Letters, February 1999, Elsevier

    Elisabeth Davioud-Charvet

  100. Evidence for the co-existence of glutathione reductase and trypanothione reductase in the non-trypanosomatid Euglenozoa: Euglena gracilis Z

    Article • FEBS Letters, January 1999, Wiley

    Elisabeth Davioud-Charvet

  101. 18-Vinyldeoxycorticosterone: a potent inhibitor of the bovine cytochrome P-45011β

    Article • Bioorganic & Medicinal Chemistry, October 1998, Elsevier

    Elisabeth Davioud-Charvet

  102. Photoaffinity labelling of the human mineralocorticoid receptor with steroids having a reactive group at position 3, 18 or 21

    Article • Biochimica et Biophysica Acta (BBA) - Protein Structure and Molecular Enzymology, October 1998, Elsevier

    Elisabeth Davioud-Charvet

  103. Structure-activity relationships in 2-aminodiphenylsulfides against trypanothione reductase from Trypanosoma cruzi

    Article • Bioorganic & Medicinal Chemistry Letters, May 1998, Elsevier

    Elisabeth Davioud-Charvet

  104. A General Approach to the Synthesis of Polyamine Linked-Monoindolylmaleimides, a New Series of Trypanothione Reductase Inhibitors.

    Article • Chemical and Pharmaceutical Bulletin, January 1998, Pharmaceutical Society of Japan

    Oleg Melnyk, Elisabeth Davioud-Charvet

  105. New spermine and spermidine derivatives as potent inhibitors of Trypanosoma cruzi Trypanothione Reductase

    Article • Bioorganic & Medicinal Chemistry, July 1997, Elsevier

    Elisabeth Davioud-Charvet

  106. Glutathione-dependent activities of Trypanosoma cruzi p52 makes it a new member of the thiol:disulphide oxidoreductase family

    Article • Biochemical Journal, February 1997, Portland Press Ltd.

    Elisabeth Davioud-Charvet

  107. New potent inhibitors of trypanothione reductase from Trypanosoma cruzi in the 2-aminodiphenylsulfide series

    Article • European Journal of Medicinal Chemistry, January 1997, Elsevier

    Elisabeth Davioud-Charvet

  108. New Steroidal Diazo Ketones as Potential Photoaffinity Labeling Reagents for the Mineralocorticoid Receptor:  Synthesis and Biological Activities

    Article • Journal of Medicinal Chemistry, January 1996, American Chemical Society (ACS)

    Elisabeth Davioud-Charvet

  109. The mineralocorticoid activity of progesterone derivatives depends on the nature of the C18 substituent.

    Article • Endocrinology, December 1995, Endocrine Society

    Dr Franck Sobrio, Elisabeth Davioud-Charvet

  110. The mineralocorticoid activity of progesterone derivatives depends on the nature of the C18 substituent

    Article • Endocrinology, December 1995, Endocrine Society

    Elisabeth Davioud-Charvet

  111. Synthesis of potential cytochrome P45011β-generated intermediates

    Article • Tetrahedron, March 1995, Elsevier

    Elisabeth Davioud-Charvet

  112. Purification of Microsomal Native Cytochrome b5 fromPotato Tubers (Solanum tuberosum L.)

    Article • Journal of Plant Physiology, January 1995, Elsevier

    Elisabeth Davioud-Charvet

  113. An improved synthesis of 18-norandrost-4-ene-3,17-dione

    Article • Steroids, March 1993, Elsevier

    Elisabeth Davioud-Charvet

  114. High Sensitivity to Auxin is a Common Feature of Hairy Root

    Article • PLANT PHYSIOLOGY, October 1990, American Society of Plant Biologists (ASPB)

    Elisabeth Davioud-Charvet

  115. Iridoid Glucosides and Phenylpropanoid Glycosides fromDeplanchea speciosa

    Article • Planta Medica, February 1989, Thieme Publishing Group

    Elisabeth Davioud-Charvet

  116. Epiallo-yohimbine derivatives isolated from in vitro hairy-root cultures of Catharanthus trichophyllus

    Article • Phytochemistry, January 1989, Elsevier

    Elisabeth Davioud-Charvet

  117. Production of indole alkaloids by in vitro root cultures from Catharanthus trichophyllus

    Article • Phytochemistry, January 1989, Elsevier

    Elisabeth Davioud-Charvet

  118. Iridoids ofRandia ruiziana

    Article • Planta Medica, February 1988, Thieme Publishing Group

    Elisabeth Davioud-Charvet

  119. Structure and Synthesis of Cucumopine, a New Crown Gall and Hairy-root Opine

    Article • Heterocycles, January 1988, Japan Institute of Heterocyclic Chemistry

    Elisabeth Davioud-Charvet

  120. Cucumopine—a new T-DNA-encoded opine in hairy root and crown gall

    Article • Phytochemistry, January 1988, Elsevier

    Elisabeth Davioud-Charvet

  121. Iridoids of Guyanese Species of Stigmaphyllon

    Article • Planta Medica, February 1985, Thieme Publishing Group

    Elisabeth Davioud-Charvet