All Stories

  1. Fluorothiazynes as SuFEx Ambiphiles: Interconversion to Amino‐sulfurdiimidoyl Fluorides

    Article • Angewandte Chemie, December 2025, Wiley

    Professor Wim M De Borggraeve

  2. Fluorothiazynes as SuFEx Ambiphiles: Interconversion to Aminosulfurdiimidoyl Fluorides

    Article • August 2025, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  3. 3D Histological Analysis of Soft Tissues by Contrast-Enhanced X-Ray Microfocus Computed Tomography: Screening and Staining Optimization of Contrast-Enhancing Staining Agents

    Article • Microscopy and Microanalysis, March 2025, Oxford University Press (OUP)

    Professor Wim M De Borggraeve

  4. Contrast-enhancing staining agents for ex vivo contrast-enhanced computed tomography: A review

    Article • Tomography of Materials and Structures, March 2025, Elsevier

    Professor Wim M De Borggraeve

  5. Enhanced decoupling of conductivity relaxation from structural relaxation in non-stoichiometric protic ionic liquids involving triflic acid and 2-aminoethyl hydrogen sulfate

    Article • The Journal of Chemical Physics, November 2024, American Institute of Physics

    Professor Wim M De Borggraeve

  6. Novel Far-Red Fluorescent 1,4-Dihydropyridines for L-Type Calcium Channel Imaging

    Article • Journal of Medicinal Chemistry, October 2024, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  7. Perfluorooxosulfate Salts as SOF4‐Gas‐Free Precursors to Multidimensional SuFEx Electrophiles

    Article • Angewandte Chemie, May 2024, Wiley

    Professor Wim M De Borggraeve

  8. Perfluorooxosulfate Salts as SOF4‐Gas‐Free Precursors to Multidimensional SuFEx Electrophiles

    Article • Angewandte Chemie, May 2024, Wiley

    Professor Wim M De Borggraeve

  9. Ex-situ ChloGen: A facile and straightforward entry to Aryl-IF4 compounds

    Article • Journal of Fluorine Chemistry, April 2024, Elsevier

    Professor Wim M De Borggraeve

  10. 1.10 The Pentafluorosulfanyl Group (SF5)

    Article • January 2024, Thieme Publishing Group

    Professor Wim M De Borggraeve

  11. An Extrusion Strategy for On-Demand SF5Cl Gas Generation from a Commercial Disulfide

    Article • Organic Letters, December 2023, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  12. Solvent‐Free Hydrohalogenation and Deuteriohalogenation by Ex Situ Generation of HX and DX Gas

    Article • European Journal of Organic Chemistry, October 2023, Wiley

    Professor Wim M De Borggraeve

  13. Charge transport in highly acidic glass-forming protic ionic liquids tailored by zwitterionic precursors

    Article • The Journal of Chemical Physics, October 2023, American Institute of Physics

    Professor Wim M De Borggraeve

  14. Polyketide Synthase‐Mediated O‐Methyloxime Formation in the Biosynthesis of the Oximidine Anticancer Agents

    Article • Angewandte Chemie, June 2023, Wiley

    Professor Wim M De Borggraeve

  15. Ex situ Generation of Thiazyl Trifluoride (NSF3) as a Gaseous SuFEx Hub**

    Article • Angewandte Chemie, June 2023, Wiley

    Professor Wim M De Borggraeve

  16. Ex situ Generation of Thiazyl Trifluoride (NSF3) as a Gaseous SuFEx Hub**

    Article • Angewandte Chemie, June 2023, Wiley

    Professor Wim M De Borggraeve

  17. Revealing the three-dimensional murine brain microstructure by contrast-enhanced computed tomography

    Article • Frontiers in Neuroscience, March 2023, Frontiers

    Professor Wim M De Borggraeve

  18. Does Supramolecular Gelation Require an External Trigger?

    Article • Gels, December 2022, MDPI AG

    Professor Wim M De Borggraeve

  19. De-risking S–F bond formation: A gas cylinder-free strategy to access S(IV) and S(VI) fluorinated compounds.

    Article • November 2022, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  20. Cryogenic contrast-enhanced microCT enables nondestructive 3D quantitative histopathology of soft biological tissues

    Article • Nature Communications, October 2022, Springer Science + Business Media

    Professor Wim M De Borggraeve

  21. 3-Methyl 5-{3-[(4-Methylbenzenesulfonyl)oxy]propyl} 4-(2,3-Dichlorophenyl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate

    Article • Molbank, October 2022, MDPI AG

    Professor Wim M De Borggraeve

  22. Chemistry of Pentafluorosulfanyl Derivatives and Related Analogs: From Synthesis to Applications

    Article • Chemistry - A European Journal, August 2022, Wiley

    Professor Wim M De Borggraeve

  23. From the North Sea to Drug Repurposing, the Antiseizure Activity of Halimide and Plinabulin

    Article • Pharmaceuticals, February 2022, MDPI AG

    Professor Wim M De Borggraeve

  24. Carbonylation Chemistry Applied to the Synthesis of Benzimidazo[2,1‐ b ]quinazolin‐12‐ones

    Article • European Journal of Organic Chemistry, January 2022, Wiley

    Professor Wim M De Borggraeve

  25. 1,3-Diazepines

    Article • January 2022, Elsevier

    Professor Wim M De Borggraeve

  26. Penicillins

    Article • January 2022, Elsevier

    Professor Wim M De Borggraeve

  27. SuFEx-enabled, chemoselective synthesis of triflates, triflamides and triflimidates

    Article • Chemical Science, January 2022, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  28. Correction: SuFEx-enabled, chemoselective synthesis of triflates, triflamides and triflimidates

    Article • Chemical Science, January 2022, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  29. Characterization of Microbial Degradation Products of Steviol Glycosides

    Article • Molecules, November 2021, MDPI AG

    Professor Wim M De Borggraeve

  30. Can the Philicity of Radicals Be Influenced by Oriented External Electric Fields?

    Article • Organic Letters, October 2021, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  31. LSA-50 paper: An alternative to P81 phosphocellulose paper for radiometric protein kinase assays

    Article • Analytical Biochemistry, October 2021, Elsevier

    Professor Wim M De Borggraeve

  32. Computational Tools to Rationalize and Predict the Self-Assembly Behavior of Supramolecular Gels

    Article • Gels, July 2021, MDPI AG

    Professor Wim M De Borggraeve

  33. Frontispiece: Lighting Up the Plasma Membrane: Development and Applications of Fluorescent Ligands for Transmembrane Proteins

    Article • Chemistry - A European Journal, June 2021, Wiley

    Professor Wim M De Borggraeve

  34. Bioassay-guided isolation of antibacterial compounds from the leaves of Tetradenia riparia with potential bactericidal effects on food-borne pathogens

    Article • Journal of Ethnopharmacology, June 2021, Elsevier

    Professor Wim M De Borggraeve

  35. Lighting Up the Plasma Membrane: Development and Applications of Fluorescent Ligands for Transmembrane Proteins

    Article • Chemistry - A European Journal, June 2021, Wiley

    Professor Wim M De Borggraeve

  36. Developments in the Discovery and Design of Protein Kinase D Inhibitors

    Article • ChemMedChem, May 2021, Wiley

    Professor Wim M De Borggraeve

  37. Copper(0) nanoparticle catalyzed Z ‐Selective Transfer Semihydrogenation of Internal Alkynes

    Article • Advanced Synthesis & Catalysis, May 2021, Wiley

    Professor Wim M De Borggraeve

  38. The presence of benzophenone in sunscreens and cosmetics containing the organic UV filter octocrylene: A laboratory study

    Article • Contact Dermatitis, April 2021, Wiley

    Professor Wim M De Borggraeve

  39. Solvent-free N-Boc deprotection by ex situ generation of hydrogen chloride gas

    Article • Organic & Biomolecular Chemistry, January 2021, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  40. Ultrasmall iron oxide nanoparticles functionalized with BODIPY derivatives as potential bimodal probes for MRI and optical imaging

    Article • Nano Select, November 2020, Wiley

    Professor Wim M De Borggraeve

  41. Design, synthesis and biological evaluation of pyrazolo[3,4-d]pyrimidine-based protein kinase D inhibitors

    Article • European Journal of Medicinal Chemistry, November 2020, Elsevier

    Professor Wim M De Borggraeve

  42. Concomitant positive patch test reactions in FreeStyle‐allergic patients sensitized to isobornyl acrylate

    Article • Contact Dermatitis, October 2020, Wiley

    Professor Wim M De Borggraeve

  43. Facile Method to Obtain Low DS β-ketoesters and Esters of Microfibrillated Cellulose

    Article • Fibers and Polymers, October 2020, Springer Science + Business Media

    Professor Wim M De Borggraeve

  44. Nematicidal Activity of Holigarna caustica (Dennst.) Oken Fruit Is Due to Linoleic Acid

    Article • Biomolecules, July 2020, MDPI AG

    Professor Wim M De Borggraeve

  45. Tuning the Properties of Polyether Alkyl Urea Derivatives as Rheology Modifiers in Cosmetic Solvents

    Article • ACS Applied Polymer Materials, June 2020, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  46. Stereoselective Reductions of 3-Substituted Cyclobutanones: A Comparison between Experiment and Theory

    Article • The Journal of Organic Chemistry, May 2020, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  47. Biofilm inhibiting properties of compounds from the leaves of Warburgia ugandensis Sprague subsp ugandensis against Candida and staphylococcal biofilms

    Article • Journal of Ethnopharmacology, February 2020, Elsevier

    Professor Wim M De Borggraeve

  48. Exploring polyoxometalates as non-destructive staining agents for contrast-enhanced microfocus computed tomography of biological tissues

    Article • Acta Biomaterialia, January 2020, Elsevier

    Professor Wim M De Borggraeve

  49. Ex situ gas generation for lab scale organic synthesis

    Article • Reaction Chemistry & Engineering, January 2020, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  50. Molecular dynamics based descriptors for predicting supramolecular gelation

    Article • Chemical Science, January 2020, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  51. Rationalising Supramolecular Hydrogelation of Bis‐Urea‐Based Gelators through a Multiscale Approach

    Article • ChemPlusChem, December 2019, Wiley

    Professor Wim M De Borggraeve

  52. Rationalising Supramolecular Hydrogelation of Bis‐Urea‐Based Gelators through a Multiscale Approach

    Article • ChemPlusChem, December 2019, Wiley

    Professor Wim M De Borggraeve

  53. Rationalising Supramolecular Hydrogelation of Bis‐Urea‐Based Gelators through a Multiscale Approach

    Article • ChemPlusChem, November 2019, Wiley

    Professor Wim M De Borggraeve

  54. Introduction of Aryl Fluorosulfates into the Realm of Catellani Reaction Substrates

    Article • The Journal of Organic Chemistry, November 2019, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  55. Green approach for the activation and functionalization of jute fibers through ball milling

    Article • Cellulose, November 2019, Springer Science + Business Media

    Professor Wim M De Borggraeve

  56. Modeling of Nanomolecular and Reticular Architectures with 6-fold Grooved, Programmable Interlocking Disks

    Article • Journal of Chemical Education, October 2019, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  57. Nanocarrier systems assembled from PEGylated hyperbranched poly(arylene oxindole)

    Article • European Polymer Journal, October 2019, Elsevier

    Professor Wim M De Borggraeve

  58. Acylated sulfonamide adenosines as potent inhibitors of the adenylate-forming enzyme superfamily

    Article • European Journal of Medicinal Chemistry, July 2019, Elsevier

    Professor Wim M De Borggraeve

  59. An Effective and Reusable Hyperbranched Polymer Immobilized Rhodium Catalyst for the Hydroformylation of Olefins

    Article • ACS Applied Polymer Materials, June 2019, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  60. Electrochemistry and Photoredox Catalysis: A Comparative Evaluation in Organic Synthesis

    Article • Molecules, June 2019, MDPI AG

    Professor Wim M De Borggraeve

  61. Ketone Synthesis by a Nickel-Catalyzed Dehydrogenative Cross-Coupling of Primary Alcohols

    Article • Journal of the American Chemical Society, April 2019, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  62. Synthesis of N-Acyl Sulfamates from Fluorosulfates and Amides

    Article • The Journal of Organic Chemistry, January 2019, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  63. Ball milling: a green technology for the preparation and functionalisation of nanocellulose derivatives

    Article • Nanoscale Advances, January 2019, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  64. Robust scalable synthesis of a bis-urea derivative forming thixotropic and cytocompatible supramolecular hydrogels

    Article • Chemical Communications, January 2019, Royal Society of Chemistry

    Professor Wim M De Borggraeve, Ramesh Subramani

  65. Chemical structure and biological properties of sulfated fucan from the sequential extraction of subAntarctic Lessonia sp (Phaeophyceae)

    Article • Carbohydrate Polymers, November 2018, Elsevier

    Professor Wim M De Borggraeve

  66. Bioassay-guided isolation of active substances from Semen Torreyae identifies two new anthelmintic compounds with novel mechanism of action

    Article • Journal of Ethnopharmacology, October 2018, Elsevier

    Professor Wim M De Borggraeve

  67. A Robust and Scalable Continuous Flow Process for Glycerol Carbonate

    Article • Chemical Engineering & Technology, September 2018, Wiley

    Professor Wim M De Borggraeve

  68. Bioassay-guided isolation of three anthelmintic compounds from Warburgia ugandensis Sprague subspecies ugandensis, and the mechanism of action of polygodial

    Article • International Journal for Parasitology, September 2018, Elsevier

    Professor Wim M De Borggraeve

  69. Identification of fukinolic acid from Cimicifuga heracleifolia and its derivatives as novel antiviral compounds against enterovirus A71 infection

    Article • International Journal of Antimicrobial Agents, July 2018, Elsevier

    Johan Neyts, Professor Wim M De Borggraeve

  70. Direct Access to Aryl Bis(trifluoromethyl)carbinols from Aryl Bromides or Fluorosulfates: Palladium-Catalyzed Carbonylation

    Article • Angewandte Chemie, May 2018, Wiley

    Professor Wim M De Borggraeve

  71. Direct Access to Aryl Bis(trifluoromethyl)carbinols from Aryl Bromides or Fluorosulfates: Palladium-Catalyzed Carbonylation

    Article • Angewandte Chemie, May 2018, Wiley

    Professor Wim M De Borggraeve

  72. Active principles of Tetradenia riparia . IV. Anthelmintic activity of 8(14),15-sandaracopimaradiene-7α,18-diol

    Article • Journal of Ethnopharmacology, April 2018, Elsevier

    Professor Wim M De Borggraeve

  73. Non-innocent probes in direct sonication: Metal assistance in oxidative radical C H functionalization

    Article • Ultrasonics Sonochemistry, March 2018, Elsevier

    Professor Wim M De Borggraeve

  74. Methylated flavonoids as anti-seizure agents: Naringenin 4′,7-dimethyl ether attenuates epileptic seizures in zebrafish and mouse models

    Article • Neurochemistry International, January 2018, Elsevier

    Professor Wim M De Borggraeve

  75. Synthesis and peptide functionalization of hyperbranched poly(arylene oxindole) towards versatile biomaterials

    Article • Polymer Chemistry, January 2018, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  76. Synthesis of an IS and Steviol Glycoside Analysis by a Validated Internal Standard Method

    Article • American Journal of Analytical Chemistry, January 2018, Scientific Research Publishing, Inc,

    Professor Wim M De Borggraeve

  77. Flow-Assisted Synthesis of Heterocycles via Multicomponent Reactions

    Article • January 2018, Springer Science + Business Media

    Professor Wim M De Borggraeve

  78. Functionalization of Heteroarenes Under Continuous Flow

    Article • January 2018, Springer Science + Business Media

    Professor Wim M De Borggraeve

  79. Water Tolerant and Reusable Sulfonated Hyperbranched Poly(aryleneoxindole) Acid Catalyst for Solvent-Free Esterification

    Article • ChemistrySelect, October 2017, Wiley

    Professor Wim M De Borggraeve

  80. Ex Situ Generation of Sulfuryl Fluoride for the Synthesis of Aryl Fluorosulfates

    Article • Organic Letters, September 2017, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  81. A Convenient Multigram Synthesis of DABSO Using Sodium Sulfite as SO2 Source

    Article • Organic Process Research & Development, April 2017, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  82. Crystal structure of 5-benzyl-8-bromo-2-methyl-1,3-oxazolo[4,5-c][1,8]naphthyridin-4(5H)-one

    Article • Acta Crystallographica Section E Crystallographic Communications, April 2017, International Union of Crystallography

    Professor Wim M De Borggraeve

  83. Towards New Tricyclic Motifs: Intramolecular C-H Arylation as the Key Step in a Formal [3+3] Cyclocondensation Strategy

    Article • European Journal of Organic Chemistry, March 2017, Wiley

    Professor Wim M De Borggraeve

  84. Intramolecular Carbonylative C-H Functionalization of 1,2,3- Triazoles for the Synthesis of Triazolo[1,5-a]indolones

    Article • Advanced Synthesis & Catalysis, February 2017, Wiley

    Professor Wim M De Borggraeve

  85. Discovery of a potent protein kinase D inhibitor: insights in the binding mode of pyrazolo[3,4-d]pyrimidine analogues

    Article • MedChemComm, January 2017, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  86. Carbonylation as a novel method for the assembly of pyrazine based oligoamide alpha-helix mimetics

    Article • Organic & Biomolecular Chemistry, January 2017, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  87. Nanocellulosic materials as bioinks for 3D bioprinting

    Article • Biomaterials Science, January 2017, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  88. The orthorhombic pseudopolymorph of tacrine hydrochloride

    Article • Acta Crystallographica Section B Structural Science Crystal Engineering and Materials, September 2016, International Union of Crystallography

    Professor Wim M De Borggraeve

  89. Low-cost instant CO generation at room temperature using formic acid, mesyl chloride and triethylamine

    Article • Reaction Chemistry & Engineering, January 2016, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  90. Gadolinium(III)-DOTA Complex Functionalized with BODIPY as a Potential Bimodal Contrast Agent for MRI and Optical Imaging

    Article • Inorganics, November 2015, MDPI AG

    Professor Wim M De Borggraeve

  91. Luminescence and Relaxometric Properties of Heteropolymetallic Metallostar Complexes with Selectively Incorporated Lanthanide(III) Ions

    Article • European Journal of Inorganic Chemistry, August 2015, Wiley

    Professor Wim M De Borggraeve

  92. Improved detection of β-N-methylamino-l-alanine using N-hydroxysuccinimide ester of N-butylnicotinic acid for the localization of BMAA in blue mussels (Mytilus edulis)

    Article • Analytical and Bioanalytical Chemistry, March 2015, Springer Science + Business Media

    Professor Wim M De Borggraeve

  93. Synthesis of N -Hydroxypyrazin-2(1 H )-ones via Selective O -Debenzylation of 1-Benzyloxypyrazin-2(1 H )-ones Using Flow Methodology

    Article • Journal of Flow Chemistry, March 2015, Akademiai Kiado

    Professor Wim M De Borggraeve

  94. First Example of Alkyl–Aryl Negishi Cross-Coupling in Flow: Mild, Efficient and Clean Introduction of Functionalized Alkyl Groups

    Article • Journal of Flow Chemistry, March 2015, Akademiai Kiado

    Professor Wim M De Borggraeve

  95. Facile azide formation via diazotransfer reaction in a copper tube flow reactor

    Article • Tetrahedron Letters, March 2015, Elsevier

    Professor Tatjana N. Parac-Vogt, Professor Wim M De Borggraeve

  96. The Zeamine Antibiotics Affect the Integrity of Bacterial Membranes

    Article • Applied and Environmental Microbiology, December 2014, ASM Journals

    Miss Joleen Masschelein, Prof Yves Briers, Professor Wim M De Borggraeve

  97. First Example of a Continuous-Flow Carbonylation Reaction Using Aryl Formates as CO Precursors

    Article • Journal of Flow Chemistry, September 2014, Akademiai Kiado

    Professor Wim M De Borggraeve, Dr Jesus Alcazar

  98. Synthesis of 1-benzyloxypyrazin-2(1H)-one derivatives

    Article • Tetrahedron Letters, August 2014, Elsevier

    Professor Wim M De Borggraeve

  99. Synthesis of 11-aza-artemisinin derivatives using the Ugi reaction and an evaluation of their antimalarial activity

    Article • Tetrahedron Letters, August 2014, Elsevier

    Dr Nguyen Thanh Le, Professor Wim M De Borggraeve

  100. Synthesis of triterpenoid triazine derivatives from allobetulone and betulonic acid with biological activities

    Article • Bioorganic & Medicinal Chemistry, July 2014, Elsevier

    Professor Wim M De Borggraeve

  101. Synthetic Protocol toward Fused Pyrazolone Derivatives via a Michael Addition and Reductive Ring Closing Strategy

    Article • The Journal of Organic Chemistry, June 2014, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  102. 8-HaloBODIPYs and Their 8-(C, N, O, S) Substituted Analogues: Solvent Dependent UV–Vis Spectroscopy, Variable Temperature NMR, Crystal Structure Determination, and Quantum Chemical Calculations

    Article • The Journal of Physical Chemistry A, March 2014, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  103. Formation of amides when other approaches have failed

    Article • Chemical Communications, January 2014, Royal Society of Chemistry

    Dr Jesus Alcazar, Professor Wim M De Borggraeve

  104. Tanshinone IIA Exhibits Anticonvulsant Activity in Zebrafish and Mouse Seizure Models

    Article • ACS Chemical Neuroscience, November 2013, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  105. Diterpene glycosides from Stevia phlebophylla A. Gray

    Article • Carbohydrate Research, September 2013, Elsevier

    Professor Wim M De Borggraeve

  106. Alpha-Helical Destabilization of the Bcl-2-BH4-Domain Peptide Abolishes Its Ability to Inhibit the IP3 Receptor

    Article • PLOS One, August 2013, PLOS

    Professor Wim M De Borggraeve, Giovanni Monaco

  107. Synthesis and in vitro evaluation of a PDT active BODIPY–NLS conjugate

    Article • Bioorganic & Medicinal Chemistry Letters, June 2013, Elsevier

    Professor Wim M De Borggraeve

  108. Asymmetric Synthesis of 1-Aza-4-deoxypicropodophyllotoxin

    Article • Synlett, April 2013, Thieme Publishing Group

    Professor Wim M De Borggraeve

  109. Scaffold Hoppingviaa Transannular Rearrangement–Encompassing Cascade

    Article • Organic Letters, February 2013, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  110. Absolute configuration of 3-acetylbetulinic acid

    Article • Journal of Structural Chemistry, February 2013, Pleiades Publishing Ltd

    Professor Wim M De Borggraeve

  111. Preparation and characterization of hydrogels based on homopolymeric fractions of sodium alginate and PNIPAAm

    Article • Carbohydrate Polymers, January 2013, Elsevier

    Professor Wim M De Borggraeve

  112. Total Synthesis of Septocylindrin B and C-Terminus Modified Analogues

    Article • PLOS One, December 2012, PLOS

    Professor Wim M De Borggraeve

  113. Fused derivatives of (iso)steviol via pericyclic reactions

    Article • Tetrahedron Letters, December 2012, Elsevier

    Professor Wim M De Borggraeve

  114. Stevioside and Steviol as Starting Materials in Organic Synthesis

    Article • Current Organic Chemistry, September 2012, Bentham Science Publishers

    Professor Wim M De Borggraeve

  115. Tetranuclear d-f Metallostars: Synthesis, Relaxometric, and Luminescent Properties

    Article • Inorganic Chemistry, July 2012, American Chemical Society (ACS)

    Professor Tatjana N. Parac-Vogt, Professor Wim M De Borggraeve

  116. A Tripodal Ruthenium–Gadolinium Metallostar as a Potential αvβ3Integrin Specific Bimodal Imaging Contrast Agent

    Article • Inorganic Chemistry, June 2012, American Chemical Society (ACS)

    Professor Tatjana N. Parac-Vogt, Professor Wim M De Borggraeve, Professor Carmen Burtea

  117. Anticonvulsant activity of bisabolene sesquiterpenoids of Curcuma longa in zebrafish and mouse seizure models

    Article • Epilepsy & Behavior, May 2012, Elsevier

    Professor Wim M De Borggraeve

  118. Selective LC-MS/MS method for the identification of BMAA from its isomers in biological samples

    Article • Analytical and Bioanalytical Chemistry, April 2012, Springer Science + Business Media

    Professor Wim M De Borggraeve

  119. Identification of a Small Molecule That Modulates Platelet Glycoprotein Ib-von Willebrand Factor Interaction

    Article • Journal of Biological Chemistry, January 2012, American Society for Biochemistry & Molecular Biology (ASBMB)

    Professor Wim M De Borggraeve

  120. An integrated fragment based screening approach for the discovery of small molecule modulators of the VWF–GPIbα interaction

    Article • Chemical Communications, January 2012, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  121. The C Terminus of Bax Inhibitor-1 Forms a Ca2+-permeable Channel Pore

    Article • Journal of Biological Chemistry, November 2011, American Society for Biochemistry & Molecular Biology (ASBMB)

    Professor Wim M De Borggraeve

  122. A Heterobimetallic Ruthenium–Gadolinium Complex as a Potential Agent for Bimodal Imaging

    Article • Inorganic Chemistry, October 2011, American Chemical Society (ACS)

    Professor Tatjana N. Parac-Vogt, Professor Wim M De Borggraeve

  123. Rational Design, Synthesis, and Spectroscopic and Photophysical Properties of a Visible-Light-Excitable, Ratiometric, Fluorescent Near-Neutral pH Indicator Based on BODIPY

    Article • Chemistry - A European Journal, August 2011, Wiley

    Professor Wim M De Borggraeve

  124. Isosteviol as a Starting Material in Organic Synthesis

    Article • Current Organic Chemistry, August 2011, Bentham Science Publishers

    Professor Wim M De Borggraeve

  125. A Modular Approach towards the Synthesis of Target-Specific MRI Contrast Agents

    Article • European Journal of Inorganic Chemistry, July 2011, Wiley

    Professor Tatjana N. Parac-Vogt, Professor Wim M De Borggraeve, Professor Carmen Burtea

  126. Synthesis of the orthogonally protected amino alcohol Phaol and analogs

    Article • Journal of Peptide Science, April 2011, Wiley

    Professor Wim M De Borggraeve

  127. 2-(4-Methoxybenzyl)-4,6-diphenyl-2,5-diazabicyclo[2.2.2]oct-5-en-3-one

    Article • Acta Crystallographica Section E Structure Reports Online, April 2011, International Union of Crystallography

    Professor Luc Van Meervelt, Professor Wim M De Borggraeve

  128. Comparison of distance information in [TOAC1, Glu(OMe)7, 18, 19] alamethicin F50/5 from paramagnetic relaxation enhancement measurements with data obtained from an X-ray diffraction-based model

    Article • Journal of Peptide Science, March 2011, Wiley

    Professor Wim M De Borggraeve

  129. Measuring cooperative Rev protein-protein interactions on Rev responsive RNA by fluorescence resonance energy transfer

    Article • RNA Biology, March 2011, Taylor & Francis

    Professor Wim M De Borggraeve

  130. ChemInform Abstract: Synthesis of Pyridodiazepinediones by Using the Ugi Multicomponent Reaction.

    Article • ChemInform, January 2011, Wiley

    Professor Wim M De Borggraeve

  131. Triple Hyp→Pro replacement in integramide A, a peptaib inhibitor of HIV‐1 integrase: Effect on conformation and bioactivity

    Article • Biopolymers, January 2011, Wiley

    Sheo Singh, Professor Wim M De Borggraeve

  132. Synthesis of Pyridodiazepinediones by Using the Ugi Multicomponent Reaction

    Article • European Journal of Organic Chemistry, August 2010, Wiley

    Professor Wim M De Borggraeve

  133. Generalized solvent scales as a tool for investigating solvent dependence of spectroscopic and kinetic parameters. Application to fluorescent BODIPY dyes

    Article • Photochemical & Photobiological Sciences, July 2010, Springer Science + Business Media

    Professor Wim M De Borggraeve

  134. Influence of Reducing Carbohydrates on (6S)-5-Methyltetrahydrofolic Acid Degradation during Thermal Treatments

    Article • Journal of Agricultural and Food Chemistry, May 2010, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  135. Direct functionalization of BODIPY dyes by oxidative nucleophilic hydrogen substitution at the 3- or 3,5-positions

    Article • Chemical Communications, January 2010, Royal Society of Chemistry

    Professor Wim M De Borggraeve

  136. Synthesis and Substitution of 8-(4,6-Dichloropyrimidin-5-yl)-BODIPY

    Article • European Journal of Organic Chemistry, December 2009, Wiley

    Professor Wim M De Borggraeve

  137. Synthesis and Biological Evaluation of Bridged Analogues of the Platelet Aggregation Inhibitor Trifenagrel

    Article • Letters in Drug Design & Discovery, October 2009, Bentham Science Publishers

    Professor Wim M De Borggraeve

  138. Flavonoids from Senecio viscosus

    Article • Chemistry of Natural Compounds, September 2009, Springer Science + Business Media

    Professor Wim M De Borggraeve

  139. Mechanism and Related Kinetics of 5-Methyltetrahydrofolic Acid Degradation during Combined High Hydrostatic Pressure−Thermal Treatments

    Article • Journal of Agricultural and Food Chemistry, August 2009, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  140. Photophysics and stability of cyano-substituted boradiazaindacene dyes

    Article • Photochemical & Photobiological Sciences, July 2009, Springer Science + Business Media

    Professor Wim M De Borggraeve

  141. Synthesis and modifications of a small library of 1,4-benzodiazepin-3-ones toward potential inhibitors of the collagen—von Willebrand Factor interaction

    Article • Tetrahedron, June 2009, Elsevier

    Professor Wim M De Borggraeve

  142. Synthesis of 5,5′-Dialkyl-6,6′-dichloro-2, 2′-bipyridines

    Article • Synthetic Communications, February 2009, Taylor & Francis

    Professor Wim M De Borggraeve

  143. ChemInform Abstract: Synthesis of Pyrazino[1,2‐a]benzimidazol‐1(2H)ones via a Microwave‐Assisted Buchwald—Hartwig Type Reaction.

    Article • ChemInform, November 2008, Wiley

    Professor Wim M De Borggraeve

  144. Structural property investigations of 1-[2-(2-methoxyphenyl)ethyl]piperidinium chloride: An experimental and computational study

    Article • Journal of Molecular Structure, November 2008, Elsevier

    Professor Wim M De Borggraeve

  145. Synthesis of Highly Functionalized 2(1H)-Pyrazinone 3-Carboxamide Scaffolds

    Article • Organic Letters, September 2008, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  146. Synthesis of pyrazino[1,2-a]benzimidazol-1(2H)ones via a microwave assisted Buchwald–Hartwig type reaction

    Article • Tetrahedron, August 2008, Elsevier

    Professor Wim M De Borggraeve

  147. Ratiometric, Fluorescent BODIPY Dye with Aza Crown Ether Functionality: Synthesis, Solvatochromism, and Metal Ion Complex Formation

    Article • The Journal of Physical Chemistry A, July 2008, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  148. Matrix-isolation FT-IR and theoretical investigation of the competitive intramolecular hydrogen bonding in 5-methyl-3-nitro-2-hydroxyacetophenone

    Article • Journal of Molecular Structure, May 2008, Elsevier

    Professor Wim M De Borggraeve

  149. Spirocyclic Pyridoazepine Analogues of Galanthamine: Synthesis, Modelling Studies and Evaluation as Inhibitors of Acetylcholinesterase

    Article • European Journal of Organic Chemistry, May 2008, Wiley

    Professor Wim M De Borggraeve

  150. ATR-IR spectroscopic study of the structural changes in the hydrophobic region of ICPAN/DPPC bilayers

    Article • Journal of Molecular Structure, April 2008, Elsevier

    Professor Wim M De Borggraeve

  151. Synthesis and Biological Evaluation of Methylene-Bridged Analogs of the Potent Cannabinoid Receptor Antagonist Rimonabant

    Article • European Journal of Organic Chemistry, March 2008, Wiley

    Professor Wim M De Borggraeve

  152. trans-Chlorido[6-chloro-4-(4-methoxybenzyl)-3-oxo-3,4-dihydropyrazin-2-yl]bis(triphenylphosphine)palladium(II)

    Article • Acta Crystallographica Section E Structure Reports Online, December 2007, International Union of Crystallography

    Professor Wim M De Borggraeve

  153. Matrix-isolation FT-IR and theoretical investigation of the vibrational properties of the sterically hindered ortho-hydroxy acylaromatic Schiff bases

    Article • Journal of Molecular Structure, November 2007, Elsevier

    Professor Wim M De Borggraeve

  154. Synthesis of Spirocyclic Pyridoazepines as Analogues of Galanthamine by Nucleophilic Aromatic Substitution of 3‐Substituted 2‐Chloropyridines

    Article • European Journal of Organic Chemistry, October 2007, Wiley

    Professor Wim M De Borggraeve

  155. Photophysics of 3,5-diphenoxy substituted BODIPY dyes in solution

    Article • Photochemical & Photobiological Sciences, October 2007, Springer Science + Business Media

    Professor Wim M De Borggraeve

  156. Synthesis of Methylene‐Bridged Analogues of Biologically Active Pteridine Derivatives.

    Article • ChemInform, September 2007, Wiley

    Professor Wim M De Borggraeve

  157. Synthesis of Methylene‐Bridged Analogues of Biologically Active Pteridine Derivatives

    Article • European Journal of Organic Chemistry, June 2007, Wiley

    Professor Wim M De Borggraeve

  158. Conformational Analysis of TOAC‐Labelled Alamethicin F50/5 Analogues

    Article • Chemistry & Biodiversity, June 2007, Wiley

    Professor Wim M De Borggraeve

  159. Design, Synthesis and Evaluation of Serine Protease Inhibitor Analogues

    Article • European Journal of Organic Chemistry, June 2007, Wiley

    Professor Wim M De Borggraeve

  160. Synthesis of 2(1H)‐Pyrazinone Phosphonates via an Arbuzov‐Type Reaction.

    Article • ChemInform, May 2007, Wiley

    Professor Wim M De Borggraeve

  161. Diastereoselective Diels—Alder Additions of Ethene to Substituted Homochiral 2(1H)‐Pyrazinones.

    Article • ChemInform, May 2007, Wiley

    Professor Wim M De Borggraeve

  162. Diastereoselective Diels–Alder Additions of Ethene to Substituted Homochiral 2(1H)-Pyrazinones

    Article • European Journal of Organic Chemistry, February 2007, Wiley

    Professor Wim M De Borggraeve

  163. Synthesis of 2(1H)-Pyrazinone Phosphonates via an Arbuzov-type Reaction

    Article • The Journal of Organic Chemistry, December 2006, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  164. 3,5‐Dihalo‐2(1H)‐pyrazinones: Versatile Scaffolds in Organic Synthesis

    Article • ChemInform, November 2006, Wiley

    Professor Wim M De Borggraeve

  165. 3,5-Dihalo-2(1 H )-pyrazinones: Versatile Scaffolds in Organic Synthesis

    Article • Synthesis, September 2006, Thieme Publishing Group

    Professor Wim M De Borggraeve

  166. Photophysical properties of an on/off fluorescent pH indicator excitable with visible light based on a borondipyrromethene-linked phenol

    Article • Journal of Photochemistry and Photobiology A Chemistry, September 2006, Elsevier

    Professor Wim M De Borggraeve

  167. Synthesis of 1,5-disubstituted 4-haloimidazoles from α-aminonitriles

    Article • Tetrahedron Letters, July 2006, Elsevier

    Professor Wim M De Borggraeve

  168. Solvent and pH Dependent Fluorescent Properties of a Dimethylaminostyryl Borondipyrromethene Dye in Solution

    Article • The Journal of Physical Chemistry A, May 2006, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  169. Design, Synthesis, and Preferred Conformation of Peptides Based on a Highly Constrained, β,β′-Diphenyl Substituted Cyclopropane α-Amino Acid

    Article • January 2006, Springer Science + Business Media

    Professor Wim M De Borggraeve

  170. Preferred 3D-Structure of Peptides Rich in a Severely Conformationally Restricted Cyclopropane Analogue of Phenylalanine

    Article • Chemistry - A European Journal, January 2006, Wiley

    Professor Wim M De Borggraeve

  171. Structure based design of simplified analogues of insect kinins

    Article • Tetrahedron, October 2005, Elsevier

    Professor Wim M De Borggraeve

  172. Development of New Amino(oxo)piperidinecarboxylate Scaffolds and Their Evaluation as -Turn Mimics

    Article • European Journal of Organic Chemistry, July 2005, Wiley

    Professor Wim M De Borggraeve

  173. BODIPY-Based Hydroxyaryl Derivatives as Fluorescent pH Probes

    Article • The Journal of Organic Chemistry, April 2005, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  174. Expanding the substitution pattern of 2(1H)-pyrazinones via Suzuki and Heck reactions

    Article • Tetrahedron, April 2005, Elsevier

    Professor Wim M De Borggraeve

  175. Synthesis of sidechain adapted β-turn mimics for modifying the C-terminus of substance P

    Article • Tetrahedron Letters, March 2005, Elsevier

    Professor Wim M De Borggraeve

  176. Turn and Helical Peptide Handedness Governed Exclusively by Side-Chain Chiral Centers

    Article • Journal of the American Chemical Society, February 2005, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  177. Synthesis of Novel Functionalised Symmetric Bi-2(1 H )-pyrazinones

    Article • Synlett, January 2005, Thieme Publishing Group

    Professor Wim M De Borggraeve

  178. Design and synthesis of novel type VI-like β-turn mimetics. Diversity at the i+1 and the i+2 position

    Article • Tetrahedron, December 2004, Elsevier

    Professor Wim M De Borggraeve

  179. New Routes for the Synthesis of 3‐ and 5‐Substituted 2(1H)‐Pyrazinones.

    Article • ChemInform, May 2004, Wiley

    Professor Wim M De Borggraeve

  180. Acid catalysed methanolysis of 2,5-diazabicyclo[2.2.2]octane-3,6-diones: scope and limitations

    Article • Tetrahedron Letters, May 2004, Elsevier

    Professor Wim M De Borggraeve

  181. New routes for the synthesis of 3- and 5-substituted 2(1H)-pyrazinones

    Article • Tetrahedron Letters, February 2004, Elsevier

    Professor Wim M De Borggraeve

  182. Stereoselective transformation of pyrazinones into substituted analogues of cis-5-amino-6-oxo-2-piperidinemethanol and cis-5-amino-2-piperidinemethanol

    Article • Tetrahedron, June 2003, Elsevier

    Professor Wim M De Borggraeve

  183. Development of a Functionalizable External β-Turn Mimic Based on a cis-Fused 1,7-Naphthyridine Scaffold

    Article • European Journal of Organic Chemistry, May 2003, Wiley

    Professor Wim M De Borggraeve

  184. High-Speed Microwave-Promoted Hetero-Diels−Alder Reactions of 2(1H)-Pyrazinones in Ionic Liquid Doped Solvents

    Article • The Journal of Organic Chemistry, November 2002, American Chemical Society (ACS)

    Professor Wim M De Borggraeve

  185. Stereoselective intramolecular Diels–Alder reactions of 3-alkenyl(oxy)-2(1H)-pyrazinones

    Article • Tetrahedron Letters, January 2002, Elsevier

    Professor Wim M De Borggraeve

  186. Intramolecular Diels–Alder reactions of N-alkenyl-2(1H)-pyrazinones: generation of a novel type of cis-1,7-naphthyridine

    Article • Tetrahedron Letters, October 2001, Elsevier

    Professor Wim M De Borggraeve

  187. Synthesis of a conformationally restricted dipeptide analogue and its evaluation as a β-turn mimic

    Article • Tetrahedron Letters, August 2001, Elsevier

    Professor Wim M De Borggraeve

  188. Divergent pathways in the intramolecular diels-alder reaction of 2(1H)-pyrazinones substituted at the 3-position with a phenylalkyne containing side chain

    Article • Tetrahedron, December 1999, Elsevier

    Professor Wim M De Borggraeve