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  1. One‐Pot Hetero‐Di‐C‐Glycosylation of the Natural Polyphenol Phloretin by a Single C‐Glycosyltransferase With Broad Sugar Substrate Specificity
  2. The novel ribosome biogenesis inhibitor usnic acid blocks nucleolar pre-60S maturation
  3. Discovery, characterization, and comparative analysis of new UGT72 and UGT84 family glycosyltransferases
  4. Klebsiella oxytoca inhibits Salmonella infection through multiple microbiota-context-dependent mechanisms
  5. Biocatalytic access to quaternary stereogenic centers using ene reductases
  6. Design, synthesis and catalytic application of water-soluble 1,1′-bis(diphenylphosphino)ferrocene ligands
  7. Loop 6 and the β‐hairpin flap are structural hotspots that determine cofactor specificity in the FMN‐dependent family of ene‐reductases
  8. Recent Advances in Pd‐Catalyzed Suzuki‐Miyaura Cross‐Coupling Reactions with Triflates or Nonaflates
  9. Constraining and Modifying Peptides Using Pd‐Mediated Cysteine Allylation
  10. Constraining and Modifying Peptides Using Pd‐Mediated Cysteine Allylation
  11. Fatty acid desaturation by stearoyl-CoA desaturase-1 controls regulatory T cell differentiation and autoimmunity
  12. Microbiota-derived genotoxin tilimycin generates colonic stem cell mutations
  13. Reaction intensification for biocatalytic production of polyphenolic natural product di‐ C ‐β‐glucosides
  14. Activity‐Based Protein Profiling of Oxidases and Reductases
  15. Enterotoxin tilimycin from gut-resident Klebsiella promotes mutational evolution and antibiotic resistance in mice
  16. Design and synthesis of efficient fluororethylene-peptidomimetic inhibitors of dipeptidyl peptidase III (DPP3)
  17. Small-Molecule Inhibitors Targeting Lipolysis in Human Adipocytes
  18. A Modular Synthesis of Teraryl‐Based α‐Helix Mimetics, Part 3: Iodophenyltriflate Core Fragments Featuring Side Chains of Proteinogenic Amino Acids
  19. A Modular Synthesis of Teraryl‐Based α‐Helix Mimetics, Part 4: Core Fragments with Two Halide Leaving Groups Featuring Side Chains of Proteinogenic Amino Acids
  20. A Modular Synthesis of Teraryl‐Based α‐Helix Mimetics, Part 5: A Complete Set of Pyridine Boronic Acid Pinacol Esters Featuring Side Chains of Proteinogenic Amino Acids
  21. Total synthesis of the isoquinolinium metabolite ETM-204 of Trabectidin
  22. Structural Changes in the Cap of Rv0183/mtbMGL Modulate the Shape of the Binding Pocket
  23. Efficient Entropy‐Driven Inhibition of Dipeptidyl Peptidase III by Hydroxyethylene Transition‐State Peptidomimetics
  24. Pharmacological inhibition of adipose tissue adipose triglyceride lipase by Atglistatin prevents catecholamine-induced myocardial damage
  25. Organische Chemie
  26. Simultaneous quantification of enterotoxins tilimycin and tilivalline in biological matrices using HPLC high resolution ESMS2 based on isotopically 15N-labeled internal standards
  27. Inhibition of ATGL in adipose tissue ameliorates isoproterenol-induced cardiac remodeling by reducing adipose tissue inflammation
  28. Synthesis of Hydrophilic Phosphorus Ligands and Their Application in Aqueous‐Phase Metal‐Catalyzed Reactions
  29. Adipose Triglyceride Lipase is needed for homeostatic control of Sterol Element-Binding Protein-1c driven hepatic lipogenesis
  30. Activity‐Based Protein Profiling (ABPP) of Oxidoreductases
  31. Structure-activity relationship studies for the development of inhibitors of murine adipose triglyceride lipase (ATGL)
  32. Stereoselective synthesis of chiral thiol-containing 1,2-aminoalcohols via SmI2-mediated coupling
  33. Synthesis of a Bcl9 Alpha-Helix Mimetic for Inhibition of PPIs by a Combination of Electrooxidative Phenol Coupling and Pd-Catalyzed Cross Coupling
  34. Organische Chemie
  35. Pd/BIPHEPHOS is an Efficient Catalyst for the Pd‐Catalyzed S ‐Allylation of Thiols with High n ‐Selectivity
  36. Labeling and Natural Post-Translational Modification of Peptides and Proteins via Chemoselective Pd-Catalyzed Prenylation of Cysteine
  37. Metabolic disease and ABHD6 alter the circulating bis(monoacylglycerol)phosphate profile in mice and humans
  38. Trendbericht Organische Chemie
  39. Synthesis of 2-Pyrrolidinones by Palladium-Catalyzed [3+2] Cycloaddition of Isocyanates
  40. Klebsiella oxytoca enterotoxins tilimycin and tilivalline have distinct host DNA-damaging and microtubule-stabilizing activities
  41. Selective Formation of 4,4′-Biphenols by Anodic Dehydrogenative Cross- and Homo-Coupling Reaction
  42. Aliphatic hydroxylation and epoxidation of capsaicin by cytochrome P450 CYP505X
  43. Atglistatin ameliorates functional decline in heart failure via adipocyte-specific inhibition of adipose triglyceride lipase
  44. Application of Threonine Aldolases for the Asymmetric Synthesis of α-Quaternary α-Amino Acids
  45. The crystal structure of monoacylglycerol lipase from M. tuberculosis reveals the basis for specific inhibition
  46. Asymmetric Reductive Carbocyclization Using Engineered Ene Reductases
  47. Asymmetrische reduktive Carbocyclisierung durch modifizierte En-Reduktasen
  48. The highlights in organic chemistry of 2017
  49. C H and C C bond insertion reactions of diazo compounds into aldehydes
  50. Synthesis of novel ligands targeting phenazine biosynthesis proteins as a strategy for antibiotic intervention
  51. Recent developments in the isolation, biological function, biosynthesis, and synthesis of phenazine natural products
  52. Biosynthesis of the Enterotoxic Pyrrolobenzodiazepine Natural Product Tilivalline
  53. Mechanisms and Specificity of Phenazine Biosynthesis Protein PhzF
  54. Erratum: Corrigendum: Pharmacological inhibition of adipose triglyceride lipase corrects high-fat diet-induced insulin resistance and hepatosteatosis in mice
  55. Pharmacological inhibition of adipose triglyceride lipase corrects high-fat diet-induced insulin resistance and hepatosteatosis in mice
  56. Highlights in organic chemistry 2016
  57. Synthesis of α,β-unsaturated aldehydes as potential substrates for bacterial luciferases
  58. Additive-Free Pd-Catalyzed α-Allylation of Imine-Containing Heterocycles
  59. Sequential and iterative Pd-catalyzed cross-coupling reactions in organic synthesis
  60. Characterization of the monolignol oxidoreductase AtBBE-like protein 15 L182V for biocatalytic applications
  61. Comparative Activity-Based Flavin-Dependent Oxidase Profiling
  62. Enzymatic hydrolysis of poly(ethylene furanoate)
  63. ChemInform Abstract: A General and Direct Reductive Amination of Aldehydes and Ketones with Electron-Deficient Anilines.
  64. Target identification of small molecule drugs and chemical probes
  65. Target identification of covalently binding drugs by activity-based protein profiling (ABPP)
  66. Tracking Protein S-Fatty Acylation with Proteomics
  67. Crystal structure of the Saccharomyces cerevisiae monoglyceride lipase Yju3p
  68. Future Directions of Modern Organic Synthesis
  69. Organic Chemistry 2015
  70. A General and Direct Reductive Amination of Aldehydes and Ketones with Electron-Deficient Anilines
  71. Aus zwei mach eins: die Biosynthese der Phenazine
  72. ChemInform Abstract: Chemical Genetic Approaches for the Investigation of Neutral Lipid Metabolism
  73. Chemical Genetic Approaches for the Investigation of Neutral Lipid Metabolism
  74. ChemInform Abstract: A Rapid and Efficient One-Pot Method for the Reduction of N-Protected α-Amino Acids to Chiral α-Amino Aldehydes Using CDI/DIBAL-H.
  75. ChemInform Abstract: A Robust and Simple Protocol for the Synthesis of Arylfluorophosphonates.
  76. Improved and scalable synthesis of building blocks for the modular synthesis of teraryl-based alpha-helix mimetics
  77. Diversity-Oriented Synthesis of a Library of Star-Shaped 2H-Imidazolines
  78. α/β Hydrolase Domain-containing 6 (ABHD6) Degrades the Late Endosomal/Lysosomal Lipid Bis(monoacylglycero)phosphate
  79. A robust and simple protocol for the synthesis of arylfluorophosphonates
  80. Reductions of Carboxylic Acids and Derivatives
  81. Expanding the threonine aldolase toolbox for the asymmetric synthesis of tertiary α-amino acids
  82. Adipose triglyceride lipase is involved in the mobilization of triglyceride and retinoid stores of hepatic stellate cells
  83. Biocatalyzed approach for the surface functionalization of poly(L-lactic acid) films using hydrolytic enzymes
  84. Structure–activity studies in the development of a hydrazone based inhibitor of adipose-triglyceride lipase (ATGL)
  85. Fatty Acid-binding Proteins Interact with Comparative Gene Identification-58 Linking Lipolysis with Lipid Ligand Shuttling
  86. Weighing the Proteasome for Covalent Modifications
  87. ChemInform Abstract: Recent Advances and Applications of Reductive Desulfurization in Organic Synthesis
  88. A rapid and efficient one-pot method for the reduction of N-protected α-amino acids to chiral α-amino aldehydes using CDI/DIBAL-H
  89. Recent advances and applications of reductive desulfurization in organic synthesis
  90. Biosynthese der Phenazine
  91. Enterotoxicity of a nonribosomal peptide causes antibiotic-associated colitis
  92. ChemInform Abstract: The Development of a Modular Synthesis of Teraryl-Based α-Helix Mimetics as Potential Inhibitors of Protein-Protein Interactions
  93. Exploring the new threonine aldolases with broad donor specificity
  94. Stereochemistry and Mechanism of Enzymatic and Non-Enzymatic Hydrolysis of Benzylicsec-Sulfate Esters
  95. Enzymes in Organic Synthesis
  96. The Development of a Modular Synthesis of Teraryl-Based α-Helix Mimetics as Potential Inhibitors of Protein–Protein Interactions
  97. Organische Chemie 2013
  98. More than just a Halogenase: Modification of Fatty Acyl Moieties by a Trifunctional Metal Enzyme
  99. Towards the synthesis of glycosylated dihydrochalcone natural products using glycosyltransferase-catalysed cascade reactions
  100. Investigation of one-enzyme systems in the ω-transaminase-catalyzed synthesis of chiral amines
  101. Development of small-molecule inhibitors targeting adipose triglyceride lipase
  102. Conformational Plasticity and Ligand Binding of Bacterial Monoacylglycerol Lipase
  103. Chemical Synthesis of Hormones, Pheromones and Other Bioregulators
  104. Racemization-Free Chemoenzymatic Peptide Synthesis Enabled by the Ruthenium-Catalyzed Synthesis of Peptide Enol EstersviaAlkyne-Addition and Subsequent Conversion Using Alcalase-Cross-Linked Enzyme Aggregates
  105. ChemInform Abstract: An Efficient Labeling Strategy of Drug Like Molecules with Functionalized Alkyl Linkers Using CH-Activation.
  106. A Modular Synthesis of Teraryl-Based α-Helix Mimetics, Part 1: Synthesis of Core Fragments with Two Electronically Differentiated Leaving Groups
  107. Investigation of the origin and synthetic application of the pseudodilution effect for Pd-catalyzed macrocyclisations in concentrated solutions with immobilized catalysts
  108. A Modular Synthesis of Teraryl-Based α-Helix Mimetics, Part 2: Synthesis of 5-Pyridine Boronic Acid Pinacol Ester Building Blocks with Amino Acid Side Chains in 3-Position
  109. Activity-Based Probes for Studying the Activity of Flavin-Dependent Oxidases and for the Protein Target Profiling of Monoamine Oxidase Inhibitors
  110. Aktivitätsbasierte Sondenmoleküle zur Untersuchung der Aktivität Flavin-abhängiger Oxidasen und zum Zielprotein-Profiling von Monoaminooxidase-Inhibitoren
  111. An efficient labeling strategy of drug like molecules with functionalized alkyl linkers using CH-activation
  112. ChemInform Abstract: The Witkop-Winterfeldt Oxidation Converts Tetrahydropyridoindoles into Pyrroloquinolones and Cinnolines by an Unprecedented Scaffold Rearrangement.
  113. ChemInform Abstract: A Simple Synthesis of Functionalized 3-Methyl-1-pyridinyl-1H-imidazolium Salts as Bidentate N-Heterocyclic-carbene Precursors and Their Application in Ir-Catalyzed Arene Borylation.
  114. The Witkop–Winterfeldt oxidation converts tetrahydropyridoindoles into pyrroloquinolones and cinnolines by an unprecedented scaffold rearrangement
  115. Activity-Based Protein Profiling for Natural Product Target Discovery
  116. ChemInform Abstract: Combinatorial Chemistry and the Synthesis of Compound Libraries
  117. A simple synthesis of functionalized 3-methyl-1-pyridinyl-1H-imidazolium salts as bidentate N-heterocyclic-carbene precursors and their application in Ir-catalyzed arene borylation
  118. ChemInform Abstract: Suzuki and Heck Reactions Catalyzed by Preformed Palladium Clusters and Palladium/Nickel Bimetallic Clusters.
  119. ChemInform Abstract: From Protein Domains to Drug Candidates - Natural Products as Guiding Principles in the Design and Synthesis of Compound Libraries.
  120. ChemInform Abstract: Solid-Phase Synthesis of Biomolecules
  121. Organische Chemie 2009
  122. Preparation of Biomolecule Microstructures and Microarrays by Thiol-ene Photoimmobilization
  123. ChemInform Abstract: Of Two Make One: The Biosynthesis of Phenazines
  124. The Active Site of an Enzyme Can Host Both Enantiomers of a Racemic Ligand Simultaneously
  125. Gleichzeitige Bindung beider Enantiomere eines racemischen Wirkstoffs durch das aktive Zentrum eines Enzyms
  126. Combinatorial Chemistry and the Synthesis of Compound Libraries
  127. Crystal Structure of PhzA/B from Burkholderia cepacia R18194 in complex with (S)-5-bromo-2-(piperidin-3-ylamino)benzoic acid
  128. Crystal Structure of PhzA/B from Burkholderia cepacia R18194 in complex with 5-bromo-2-((1S,3R)-3-carboxycyclohexylamino)benzoic acid
  129. Crystal Structure of PhzA/B from Burkholderia cepacia R18194 cocrystallized with 2 mM racemic 5-bromo-2-(piperidin-3-ylamino)benzoic acid
  130. Crystal Structure of PhzA/B from Burkholderia cepacia R18194 in complex with (R)-5-bromo-2-(piperidin-3-ylamino)benzoic acid
  131. Crystal Structure of PhzA/B from Burkholderia cepacia R18194 in simultaneous complex with racemic 5-bromo-2-(piperidin-3-ylamino)benzoic acid
  132. ChemInform Abstract: An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides.
  133. Of Two Make One: The Biosynthesis of Phenazines
  134. Polystyrene Sulfonyl Chloride: A Highly Orthogonal Linker Resin for the Synthesis of Nitrogen-Containing Heterocycles
  135. Polystyrolsulfonylchlorid - ein hochorthogonales Linkerharz für die Synthese von Stickstoffheterocyclen
  136. The Power of Functional Resins in Organic Synthesis.Herausgegeben von Judit Tulla-Puche und Fernando Albericio.
  137. The Power of Functional Resins in Organic Synthesis.Edited by Judit Tulla-Puche and Fernando Albericio.
  138. Classics in Stereoselective Synthesis
  139. An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides
  140. Organische Chemie 2008
  141. Crystal structure of phenazine biosynthesis protein PhzA/B from Burkholderia cepacia R18194, apo form
  142. Crystal structure of phenazine biosynthesis protein PhzA/B from Burkholderia cepacia R18194, complex with 2-(cyclohexylamino)benzoic acid
  143. Crystal structure of PhzA/B from Burkholderia cepacia R18194 crystallized in C2221
  144. ChemInform Abstract: Combinatorial Solid-Phase Natural Product Chemistry
  145. PhzA/B Catalyzes the Formation of the Tricycle in Phenazine Biosynthesis
  146. Photochemical Surface Patterning by the Thiol-Ene Reaction
  147. Photochemical Surface Patterning by the Thiol-Ene Reaction
  148. Solid-Phase Synthesis of Biomolecules
  149. The Synthetic Organic Chemist’s Companion
  150. ChemInform Abstract: The Witkop-Winterfeldt Oxidation of Indoles
  151. The Way of Synthesis: Evolution of Design and Methods for Natural Products
  152. Electrons as a Reagent in Solid-Phase Organic Synthesis
  153. A Microarray Strategy for Mapping the Substrate Specificity of Protein Tyrosine Phosphatase
  154. Eine Mikroarray-Strategie zur Untersuchung der Substratspezifitäten von Protein-Tyrosin-Phosphatasen
  155. Organic Reactions in Water: Principles, Strategies and Applications
  156. Electrons as a Reagent in Solid-Phase Organic Synthesis (Eur. J. Org. Chem. 26/2007)
  157. Electrons as a Reagent in Solid‐Phase Organic Synthesis
  158. The Investigation of Organic Reactions and their Mechanisms
  159. Organische Chemie 2006
  160. Domino Reactions in Organic Synthesis
  161. The Witkop-Winterfeldt-Oxidation of Indoles
  162. Combinatorial Chemistry - From Theory to Application (Methods and Principles in Medicinal Chemistry, Vol. 26)
  163. A generic building block for C- and N-terminal protein-labeling and protein-immobilization
  164. Electroorganic Reductions Syntheses
  165. High-Throughput Screening in Chemical Catalysis - Technologies, Strategies and Applications
  166. Homogeneous Polymer-Supported Synthesis of N-Substituted Pyrroles
  167. Organische Chemie 2005
  168. Site-Selective Protein Immobilization by Staudinger Ligation
  169. Site-Selective Protein Immobilization by Staudinger Ligation
  170. Electrolysis as an Efficient Key Step in the Homogeneous Polymer-Supported Synthesis of N-Substituted Pyrroles
  171. Evaluation of Enzyme Inhibitors in Drug Discovery. Von Robert A. Copeland.
  172. Evaluation of Enzyme Inhibitors in Drug Discovery. By Robert A. Copeland.
  173. Solid-Supported Reagents and Catalysts for the Preparation of Large Ring Compounds
  174. Nutzen und Gefahren der Biotechnologie: Liebling, Du hast die Katze geklont. Von Reinhard Renneberg, Manfred Bofinger, Jens Reich. Wiley-VCH, Weinheim 2004.260 Seiten, geb., 24,90 Euro. ISBN 3-527-31075-4
  175. Electroorganic Synthesis of 2,5-Dialkoxydihydrofurans and Pyridazines on Solid Phase Using Polymer Beads as Supports
  176. Solid-supported reagents and catalysts for the preparation of large ring compounds
  177. Preface
  178. The Staudinger Ligation — A Gift to Chemical Biology
  179. Polymer-Supported Synthesis of Non-Oligomeric Natural Products
  180. Molecular Biology in Medicinal Chemistry. Band 21 der Reihe Methods and Principles in Medicinal Chemistry. Herausgegeben von Theodor Dingermann, Dieter Steinhilber und Gerd Folkers.
  181. Molecular Biology in Medicinal Chemistry. (Series: Methods and Principles in Medicinal Chemistry, Vol. 21.) Edited by Theodor Dingermann, Dieter Steinhilber and Gerd Folkers.
  182. The Staudinger Ligation—A Gift to Chemical Biology
  183. Die Staudinger-Ligation– ein Geschenk für die Chemische Biologie
  184. Der Gipfel der Stereochemie: Bürgenstock 2004
  185. The Peak of Stereochemistry: Bürgenstock 2004
  186. Electroorganic Synthesis on the Solid Phase using Polymer Beads as Supports
  187. Elektroorganische Synthese an der festen Phase mit Polymerkügelchen als Trägermaterial
  188. An efficient and inexpensive scavenger resin for Grubbs’ catalyst
  189. Small Molecule Arrays
  190. Staudinger Ligation: A New Immobilization Strategy for the Preparation of Small-Molecule Arrays
  191. Staudinger-Ligation: eine Immobilisierungsstrategie zur Herstellung von Wirkstoff-Arrays
  192. Azide-Alkyne Coupling: A Powerful Reaction for Bioconjugate Chemistry
  193. An Easily Accessible Resin-Supported Palladium Catalyst for Sonogashira Coupling.
  194. Die chemische Genetik entdeckt das (Zebra-)Fischen
  195. Chemical Genetics Goes (Zebra) Fishing
  196. Protein Structure Similarity as Guiding Principle for Combinatorial Library Design
  197. Polymer‐Supported Synthesis of Non‐Oligomeric Natural Products
  198. An Easily Accessible Resin-SupportedPalladium Catalyst for Sonogashira Coupling
  199. Natural Product Guided Compound Library Development
  200. Book Review: Handbook of Combinatorial Chemistry. Vols. 1+2. By Kyriacos C. Nicolaou, R. Hanko and W. Hartwig
  201. Buchbesprechung: Handbook of Combinatorial Chemistry. Band 1+2. Herausgegeben von Kyriacos C. Nicolaou, R. Hanko und W. Hartwig
  202. From Protein Domains to Drug Candidates—Natural Products as Guiding Principles in the Design and Synthesis of Compound Libraries
  203. Von Proteindomänen zu Wirkstoffkandidaten – Naturstoffe als Leitstrukturen für das Design und die Synthese von Substanzbibliotheken
  204. Nachwuchswissenschaftler-Symposium Bioorganische Chemie
  205. Web Site: Lehrbücher mit Websites
  206. Web Site: Lehrbücher mit Websites
  207. Web Site: Companion Sites for Textbooks
  208. Web Site: Companion Sites for Textbooks
  209. Essentials of Biological Chemistry. Von Lorraine Buckberry und Paul Teesdale
  210. Essentials of Biological Chemistry. By Lorraine Buckberry and Paul Teesdale
  211. Size-Selective Electrochemical Preparation of Surfactant-Stabilized Pd-, Ni- and Pt/Pd Colloids
  212. Organische Chemie der Carbonylverbindungen: Modern Carbonyl Chemistry. Hrsg. von Junzo Otera. Wiley-VCH, Weinheim, 2000. 613 5., geb., 298,- DM. ISBN 3-527-29871-1
  213. Cooperative Asymmetric Catalysis with Dendrimeric [Co(salen)] Complexes
  214. Cooperative Asymmetric Catalysis with Dendrimeric [Co(salen)] Complexes
  215. POLYMER CHEMISTRY:Nickel Comes Full Cycle
  216. Nanostructured nickel-clusters as catalysts in [3+2]cycloaddition reactions
  217. Suzuki and Heck reactions catalyzed by preformed palladium clusters and bimetallic clusters
  218. A New Strategy in Heterogeneous Catalysis: The Design of Cortex Catalysts
  219. Eine neue Strategie in der heterogenen Katalyse: das Design von Cortex-Katalysatoren
  220. Polymer-Supported Synthesis of Non-Oligomeric Natural Products
  221. Reverse Chemical Genetics– An Important Strategy for the Study of Protein Function in Chemical Biology and Drug Discovery
  222. Combinatorial Solid-Phase Natural Product Chemistry