Publication
The Discovery of I-BET726 (GSK1324726A), a Potent Tetrahydroquinoline ApoA1 Up-Regulator and Selective BET Bromodomain Inhibitor
Emmanuel H. Demont, Rejbinder Kaur, Antonia J. Lewis, Mark B. Schilling, Peter E. Soden, Simon Taylor, Ann L. Walker, Matthew D. Walker, Rab K. Prinjha, Edwige Nicodème, Romain Gosmini, Van Loc Nguyen, Jérôme Toum, Christophe Simon, Jean-Marie G. Brusq, Gael Krysa, Olivier Mirguet, Alizon M. Riou-Eymard, Eric V. Boursier, Lionel Trottet, Paul Bamborough, Hugh Clark, Chun-wa Chung, Leanne Cutler
Journal of Medicinal Chemistry, October 2014, American Chemical Society (ACS)
DOI: 10.1021/jm5010539