Publication
Selective Inhibition of Bruton’s Tyrosine Kinase by a Designed Covalent Ligand Leads to Potent Therapeutic Efficacy in Blood Cancers Relative to Clinically Used Inhibitors
Bárbara B. Sousa, Cátia Rebelo de Almeida, Ana F. Barahona, Raquel Lopes, Ana Martins-Logrado, Marco Cavaco, Vera Neves, Luís A. R. Carvalho, Carlos Labão-Almeida, Ana R. Coelho, Marta Leal Bento, Ricardo M. R. M. Lopes, Bruno L. Oliveira, Miguel A. R. B. Castanho, Peter Neumeister, Alexander Deutsch, Gregory I. Vladimer, Nikolaus Krall, Cristina João, Francisco Corzana, João D. Seixas, Rita Fior, Gonçalo J. L. Bernardes
ACS Pharmacology & Translational Science, November 2022, American Chemical Society (ACS)
DOI: 10.1021/acsptsci.2c00163