Publication
Achieving In Vivo Target Depletion through the Discovery and Optimization of Benzimidazolone BCL6 Degraders
Benjamin R. Bellenie, Kwai-Ming J. Cheung, Ana Varela, Olivier A. Pierrat, Gavin W. Collie, Gary M. Box, Michael D. Bright, Sharon Gowan, Angela Hayes, Matthew J. Rodrigues, Kartika N. Shetty, Michael Carter, Owen A. Davis, Alan T. Henley, Paolo Innocenti, Louise D. Johnson, Manjuan Liu, Selby de Klerk, Yann-Vaï Le Bihan, Matthew G. Lloyd, P. Craig McAndrew, Erald Shehu, Rachel Talbot, Hannah L. Woodward, Rosemary Burke, Vladimir Kirkin, Rob L. M. van Montfort, Florence I. Raynaud, Olivia W. Rossanese, Swen Hoelder
Journal of Medicinal Chemistry, April 2020, American Chemical Society (ACS)
DOI: 10.1021/acs.jmedchem.9b02076