Publication
Optimization of a Novel Binding Motif to ( E )-3-(3,5-Difluoro-4-((1 R ,3 R )-2-(2-fluoro-2-methylpropyl)-3-methyl-2,3,4,9-tetrahydro-1 H -pyrido[3,4- b ]indol-1-yl)phenyl)acrylic Acid (AZD9496), a Potent and Orally Bioavailable Selective Estrogen Rec...
Chris De Savi, Robert H. Bradbury, Alfred A. Rabow, Richard A. Norman, Camila de Almeida, David M. Andrews, Peter Ballard, David Buttar, Rowena J. Callis, Gordon S. Currie, Jon O. Curwen, Chris D. Davies, Craig S. Donald, Lyman J. L. Feron, Helen Gingell, Steven C. Glossop, Barry R. Hayter, Syeed Hussain, Galith Karoutchi, Scott G. Lamont, Philip MacFaul, Thomas A. Moss, Stuart E. Pearson, Michael Tonge, Graeme E. Walker, Hazel M. Weir, Zena Wilson
Journal of Medicinal Chemistry, October 2015, American Chemical Society (ACS)
DOI: 10.1021/acs.jmedchem.5b00984