Publication
Identification of a novel series of BET family bromodomain inhibitors: Binding mode and profile of I-BET151 (GSK1210151A)
Jonathan Seal, Yann Lamotte, Frédéric Donche, Anne Bouillot, Olivier Mirguet, Françoise Gellibert, Edwige Nicodeme, Gael Krysa, Jorge Kirilovsky, Soren Beinke, Scott McCleary, Inma Rioja, Paul Bamborough, Chun-Wa Chung, Laurie Gordon, Toni Lewis, Ann L. Walker, Leanne Cutler, David Lugo, David M. Wilson, Jason Witherington, Kevin Lee, Rab K. Prinjha
Bioorganic & Medicinal Chemistry Letters, April 2012, Elsevier
DOI: 10.1016/j.bmcl.2012.02.041