All Stories

  1. doi.org/10.1016/j.bmc.2019.115236
  2. Synthesis of obeticholic acid, a farnesoid X receptor agonist, and its major metabolites labeled with deuterium
  3. An efficient and facile synthesis of deuterium-labeled anticancer agent bendamustine hydrochloride
  4. An efficient synthesis of deuterium-labeled degarelix acetate, a third-generation gonadotropin-releasing hormone receptor antagonist
  5. Synthesis and identification of silicon-containing HCV NS5A inhibitors
  6. Preparation of tritium-labeled PF-622, a novel fatty acid amide hydrolase inhibitor
  7. An efficient synthesis of isotope-labeled PD0331179 and its labeled metabolite
  8. Efficient syntheses of dual radioisotope-labelled PF-00217830, a D2-partial agonist for the treatment of schizophrenia disorder
  9. Asymmetric syntheses of radioactive and stable isotope-labeled β-amino acids
  10. Facile syntheses of isotope-labeled chiral octahydroindole-2-carboxylic acid and its N-methyl analog
  11. Use of an Iridium-Catalyzed Redox-Neutral Alcohol-Amine Coupling on Kilogram Scale for the Synthesis of a GlyT1 Inhibitor
  12. Syntheses of dual-radioisotope-labeled CP-I, a GABAA receptor partial agonist
  13. Efficient syntheses of isotopically labeled PD0198961, a novel synthetic coagulation factor Xa inhibitor
  14. The preparation of carbon-14 and tritium radio-labeled PD-72953
  15. Convergent syntheses of carbon-13 labeled midazolam and 1′-hydroxymidazolam
  16. Syntheses of [14C] and [2H4]PD0205520, an inhibitor of the tyrosine kinase activity of the epidermal growth factor receptor
  17. Syntheses of stable-isotope labeled [M+7] and [M+6] 2-(methylamino)imidazole
  18. Synthesis of 5,5‐dimethyl‐1‐pyrroline‐N‐oxide‐2‐14C
  19. Synthesis of 5,5-dimethyl-1-pyrroline-N-oxide-2-14C
  20. Syntheses of N-t-butyl-?-phenylnitrone-?-14C and ?-(4-pyridyl-1-oxide)-N-t-butylnitrone-?-14C
  21. Synthesis of14C-labeled S-(-)-1-phenylethylamine and its application to the synthesis of [14C] CI-1021, a potential antiemetic agent (1)
  22. Reactivity and Diastereoselectivity in the Thermal and Lewis Acid-Catalyzed Diels−Alder Reactions ofN-Sulfinylphosphoramidates1
  23. A new synthesis of (Z)-coniferyl alcohol, and characterization of its derived synthetic lignin