All Stories

  1. NHC-Catalyzed Umpolung Driven Intramolecular Cyclizations for the Generation of 3,4-Cycloheptanone Annulated Tetracyclic Indole Derivatives
  2. Benzothiazolo-quinazoline Congeners Function as Anti-microtubule Agents Triggering Mitotic Arrest in Cancer Cells
  3. NHC-Catalyzed Formal [4 + 2] Annulation of o-Formyl-Tethered Michael Acceptors and Ynones to Access Highly Functionalized Naphthalene Derivatives
  4. Carbene-Catalyzed Tandem Imine Umpolung–Intramolecular Aza-Conjugate Addition–Oxidation to Access N-Substituted Isoindolinones
  5. Photocatalyzed Energy Transfer for Atom Economical Synthesis of O‐Bridged Tricyclo‐Fused Cyclopropane Derivatives
  6. Copper‐Catalyzed Intramolecular SEAr Reaction–Oxidation under Aerobic Conditions: Synthesis of Styryl‐/Alkenyl‐Substituted Xanthone Derivatives
  7. Diaryl ether derivative inhibits GPX4 expression levels to induce ferroptosis in thyroid cancer cells
  8. Total Syntheses of h5‐HT2A Receptor Antagonist, FPTase Inhibitor, FGIN‐1‐27 and its Analog by Exploiting NHC‐Catalyzed Imine Umpolung as Key Step
  9. Design and development of intramolecular doubly vinylogous Michael addition to access 3-aryl substituted 2-alkenyl-benzofurans and -indoles
  10. Tandem Copper(I)‐Catalyzed N‐Arylation–1,4‐Conjugate Addition to Access Tetrahydroacridinones
  11. Recent Advances on the Development of Synthetic Strategies to Access Dibenzoxepine Derivatives
  12. Sequential One-Pot Carbene-Catalyzed Intramolecular Stetter Reaction and Acid-Mediated Condensation: Access to Heteroatom Analogues of π-Extended Polyaromatic Hydrocarbons
  13. Recent advances in the tandem copper-catalyzed Ullmann–GoldbergN-arylation–cyclization strategies
  14. N-Heterocyclic carbene (NHC)-catalyzed oxidation of unactivated aldimines to amides via imine umpolung under aerobic conditions
  15. Tandem aza-Michael addition–vinylogous aldol condensation: synthesis of N-bridged pyridine fused quinolones
  16. N‐Heterocyclic Carbene (NHC)‐Catalyzed Intramolecular Stetter Reaction to Access Dibenzo‐fused Seven‐membered Heterocycles
  17. Design and application of intramolecular vinylogous Michael reaction for the construction of 2-alkenyl indoles
  18. N-Heterocyclic carbene (NHC)-catalyzed intramolecular benzoin condensation–oxidation
  19. Ruthenium Catalyzed Regioselective β‐C(sp3)−H Functionalization of N‐Alkyl‐N′‐p–nitrophenyl Substituted Piperazines using Aldehydes as Alkylating Agents
  20. Tandem Copper-Catalyzed Regioselective N-Arylation–Aza-Michael Addition: Synthesis of Tetracyclic 5H-Benzothiazolo[3,2-a]quinazoline Derivatives
  21. Direct Access to (±)‐10‐Desbromoarborescidine A from Tryptamine and Pentane‐1,5‐diol
  22. N-Heterocyclic carbene (NHC)-catalyzed tandem imine umpolung–aza-Michael addition–oxidation of β-carboline cyclic imines
  23. Substrate controlled, regioselective carbopalladation for the one-pot synthesis of C4-substituted tetrahydroisoquinoline analogues
  24. One-Pot Allylation–Intramolecular Vinylogous Michael Addition–Isomerization Cascade ofo-Hydroxycinnamates and Congeners: Synthesis of Substituted Benzofuran Derivatives
  25. The base-free van Leusen reaction of cyclic imines on water: synthesis of N-fused imidazo 6,11-dihydro β-carboline derivatives
  26. Synthesis and Functionalization of N-Heterocycles Using Transition Metal-Free Cross-Dehydrogenative Coupling (CDC) Approaches
  27. Tandem Aza Michael Addition–Vinylogous Nitroaldol Condensation: Construction of Highly Substituted N-Fused 3-Nitropyrazolopyridines
  28. Ruthenium Phosphine–Pyridone Catalyzed Cross-Coupling of Alcohols To form α-Alkylated Ketones
  29. Copper-Catalyzed Tandem O-Arylation–Oxidative Cross Coupling: Synthesis of Chromone Fused Pyrazoles
  30. N-Heterocyclic carbene (NHC)-catalysed atom economical construction of 2,3-disubstituted indoles
  31. Ruthenium catalyzed β-C(sp3)–H functionalization on the ‘privileged’ piperazine nucleus
  32. Phosphine-pyridonate ligands containing octahedral ruthenium complexes: access to esters and formic acid
  33. Synthesis of Tetracyclic Tetrahydro-β-carbolines by Acid-Promoted One-Pot Sequential Formation of C−C and C−N Bonds
  34. ChemInform Abstract: Tandem Copper-Catalyzed N-Arylation-Condensation and van Leusen Reaction: Synthesis of 1,4-Benzodiazepines and Imidazobenzodiazepines (ImBDs).
  35. ChemInform Abstract: Gold(III)-Catalyzed Synthesis of Aroylbenzo[b]oxepin-3-ones from ortho-O-Propargyl-1-one Substituted Arylaldehydes.
  36. Tandem Copper-CatalyzedN-Arylation-Condensation and van Leusen Reaction: Synthesis of 1,4-Benzodiazepines and Imidazobenzodiazepines (ImBDs)
  37. ChemInform Abstract: Catalytic Enantioselective Addition of Isocyanoacetate to 3-Methyl-4-nitro-5-styrylisoxazoles under Phase Transfer Catalysis Conditions.
  38. ChemInform Abstract: Gold-Catalyzed Intramolecular Cyclization of N-Propargylic β-Enaminones for the Synthesis of 1,4-Oxazepine Derivatives.
  39. Gold(iii)-catalyzed synthesis of aroylbenzo[b]oxepin-3-ones from ortho-O-propargyl-1-one substituted arylaldehydes
  40. Acetals from primary alcohols with the use of tridentate proton responsive phosphinepyridonate iridium catalysts
  41. ChemInform Abstract: Tandem Copper (Cu) Catalyzed N-Arylation-Vinylogous Nitroaldol Condensation of 3,5-Disubstituted 4-Nitropyrazoles.
  42. Gold-Catalyzed Intramolecular Cyclization of N-Propargylic β-Enaminones for the Synthesis of 1,4-Oxazepine Derivatives
  43. ChemInform Abstract: Reaction of β-Enaminones and Acetylene Dicarboxylates: Synthesis of Substituted 1,2-Dihydropyridinones.
  44. Reaction of β-enaminones and acetylene dicarboxylates: synthesis of substituted 1,2-dihydropyridinones
  45. Tandem Copper Catalysed N-Arylation Vinylogous Nitroaldol: Synthesis of N-Fused Pyrazole Quinoline
  46. Catalytic enantioselective addition of isocyanoacetate to 3-methyl-4-nitro-5-styrylisoxazoles under phase transfer catalysis conditions
  47. ChemInform Abstract: Reaction of N-Propargylic β-Enaminones with Acetylene Dicarboxylates: Catalyst-Free Synthesis of 3-Azabicyclo[4.1.0]hepta-2,4-dienes.
  48. ChemInform Abstract: Gold-Catalyzed Cyclization of N-Propargylic β-Enaminones to Form 3-Methylene-1-pyrroline Derivatives.
  49. Gold-catalysed cyclisation of N-propargylic β-enaminones to form 3-methylene-1-pyrroline derivatives
  50. Reaction of N-propargylic β-enaminones with acetylene dicarboxylates: catalyst-free synthesis of 3-azabicyclo[4.1.0]hepta-2,4-dienes
  51. DXR Inhibition by Potent Mono- and Disubstituted Fosmidomycin Analogues
  52. Convenient Methods for the Synthesis of Chiral Amino Alcohols and Amines
  53. Synthesis of antimalarial compounds fosmidomycin and FR900098 through N- or P-alkylation reactions
  54. ChemInform Abstract: N-Heterocyclic Carbene Catalyzed Homoenolate Addition to 3-Methyl-4-nitro-5-styrylisoxazoles.
  55. N-heterocyclic carbene catalysed homoenolate addition to 3-methyl-4-nitro-5-styrylisoxazoles
  56. ChemInform Abstract: Two Tandem Sequential Reactions Catalyzed by [Au], N-Heterocyclic Carbenes (NHC) and Organic Bases.
  57. Substitution of the phosphonic acid and hydroxamic acid functionalities of the DXR inhibitor FR900098: An attempt to improve the activity against Mycobacterium tuberculosis
  58. Two tandem sequential reactions catalyzed by [Au], N-heterocyclic carbenes (NHC) and organic bases
  59. Design, Synthesis, and X-ray Crystallographic Studies of α-Aryl Substituted Fosmidomycin Analogues as Inhibitors ofMycobacterium tuberculosis1-Deoxy-d-xylulose 5-Phosphate Reductoisomerase
  60. ChemInform Abstract: Intramolecular Coupling of Chiral Diimines Using Low-Valent Titanium Reagents: Stereoselective Synthesis of Chiral 3,4-Disubstituted-2,5-diazabicyclo[4.4.0]decanes.
  61. ChemInform Abstract: Catalytic Asymmetric Conjugate Addition of Nitroalkanes to 4-Nitro-5-styrylisoxazoles.
  62. ChemInform Abstract: Catalytic Asymmetric Conjugate Addition of Nitroalkanes to 4-Nitro-5-styrylisoxazoles.
  63. TiCl4 promoted menthyl ester chiral auxiliary mediated synthesis of chiral syn-β-amino esters and applications of a representative syn-β-amino ester
  64. Catalytic Asymmetric Conjugate Addition of Nitroalkanes to 4-Nitro-5-styrylisoxazoles
  65. Catalytic Asymmetric Conjugate Addition of Nitroalkanes to 4-Nitro-5-styrylisoxazoles
  66. ChemInform Abstract: Reaction of 5-(1-Bromo-2-aryl-vinyl)-3-methyl-4-nitro-isoxazoles and 1,3-Dicarbonyl Compounds.
  67. Reaction of 5-(1-bromo-2-aryl-vinyl)-3-methyl-4-nitro-isoxazoles and 1,3-dicarbonyl compounds
  68. ChemInform Abstract: Vinylogous Nitroaldol (Henry) Reaction Using 3,5-Diethyl-4-nitroisoxazole and Carbonyl Compounds.
  69. ChemInform Abstract: Aziridination of 3-Methyl-4-nitro-5-styrylisoxazoles.
  70. Vinylogous nitroaldol (Henry) reaction using 3,5-diethyl-4-nitroisoxazole and carbonyl compounds
  71. Aziridination of 3-methyl-4-nitro-5-styrylisoxazoles
  72. Synthesis of 3-Substituted Coumarins from 2-(Acyloxy)arylaldehydes Using the TiCl4/R3N Reagent System.
  73. Synthesis of 3-substituted coumarins from 2-(acyloxy)arylaldehydes using the TiCl4/R3N reagent system
  74. Addition of Titanium Ester Enolates to Aldimines Containing a Chiral α-Methylbenzylamine Moiety: Synthesis of Chiral syn-β-Amino Esters.
  75. Addition of titanium ester enolates to aldimines containing a chiral α-methylbenzylamine moiety: synthesis of chiral syn-β-amino esters
  76. Stereoselective Synthesis of syn-β-Amino Esters Using the TiCl4/R3N Reagent System.
  77. Stereoselective synthesis of syn-β-amino esters using the TiCl4/R3N reagent system
  78. Synthesis of cis-2-Aryl-3-pyrrolidine Carboxylic Esters via Diastereoselective Cyclization of γ-Imino Esters Using a TiCl4/Et3N Reagent System.
  79. Synthesis of cis-2-aryl-3-pyrrolidine carboxylic esters via diastereoselective cyclization of γ-imino esters using a TiCl4/Et3N reagent system
  80. Intramolecular coupling of chiral diimines using low-valent titanium reagents: stereoselective synthesis of chiral 3,4-disubstituted-2,5-diazabicyclo[4.4.0]decanes