All Stories

  1. The Ireland–Claisen rearrangement strategy towards the synthesis of the schizophrenia drug, (+)-asenapine
  2. Total synthesis of a thromboxane receptor antagonist, terutroban
  3. Convergent synthesis of fully functionalized decalin skeleton of (+)-fusarisetin A
  4. Scalable synthesis of the unusual amino acid segment (ADMOA unit) of marine anti-inflammatory peptide: solomonamide A
  5. “Pruning of biomolecules and natural products (PBNP)”: an innovative paradigm in drug discovery
  6. ChemInform Abstract: Asymmetric Synthesis of C11‐C23 Fragment of Pladienolide B (I).
  7. Synthesis of the Southern Tripeptide (C1–N12) of Sanglifehrins Using Asymmetric Organocatalysis
  8. Multicomponent reactions in PEG-400: ruthenium-catalyzed synthesis of substituted pyrroles
  9. AZT-prolinamide: the nucleoside derived pyrrolidine catalysts for asymmetric aldol reactions using water as solvent
  10. Asymmetric Formal Synthesis of (+)‐Lactacystin
  11. ChemInform Abstract: Total Syntheses of Arenamides A, B and C.
  12. ChemInform Abstract: Studies Towards 1,3-Diol Units Starting from syn β-Hydroxy Acylsilanes.
  13. ChemInform Abstract: Total Synthesis of (‐)‐Seimatopolide A.
  14. 5-epi-Torrubiellutin C shows antiproliferative activity on DU145 prostate cancer cells through inactivation of the AKT/mTOR pathway
  15. ChemInform Abstract: New β‐Hydroxy Acylsilane‐Derived Building Blocks and Their Use in the Synthesis of Oxygen‐Containing Heterocycles.
  16. ChemInform Abstract: Total Syntheses of Isomeric Spiroacetal Marine Natural Products Attenols A and B.
  17. Total syntheses of arenamides A, B and C
  18. Peptidomimetic organocatalysts: efficient Michael addition of ketones onto nitroolefins with very low catalyst loading
  19. Studies towards 1,3-diol units starting from syn β-hydroxy acylsilanes
  20. Total synthesis of (−)-seimatopolide A
  21. Formation of Periodic γ‐Turns in α/β‐Hybrid Peptides: DFT and NMR Experimental Evidence
  22. ChemInform Abstract: Ruthenium‐Catalyzed Benzimidazoisoquinoline Synthesis via Oxidative Coupling of 2‐Arylbenzimidazoles with Alkynes.
  23. New β-Hydroxy Acylsilane-Derived Building Blocks and Their Use in the Synthesis of Oxygen-Containing Heterocycles
  24. Total Syntheses of Isomeric Spiroacetal Marine Natural Products Attenols A and B
  25. Synthesis of 1,4,5-Trisubstituted 1,2,3-Triazoles Amicable for Automation
  26. Ruthenium-catalyzed benzimidazoisoquinoline synthesis via oxidative coupling of 2-arylbenzimidazoles with alkynes
  27. ChemInform Abstract: Synthesis of Acylsilanes via Nickel‐Catalyzed Reactions of α‐Hydroxyallylsilanes.
  28. Synthesis of Stachybotrin C and All of Its Stereoisomers: Structure Revision
  29. Towards solomonamide A: asymmetric synthesis of the unusual γ-amino acid part
  30. Synthesis of Acylsilanes via Nickel-Catalyzed Reactions of α-Hydroxyallylsilanes
  31. ChemInform Abstract: Total Synthesis of Gabosines.
  32. Total Synthesis of (−)-α-Kainic acid via Chirality Transfer through Ireland–Claisen Rearrangement
  33. ChemInform Abstract: A Ligand‐Free Copper(II)‐Catalyzed Three‐Component Reaction in Poly(ethylene glycol) Medium: A Versatile Protocol for the Preparation of Selected 3‐Indole Derivatives.
  34. Total synthesis of 5-epi-Torrubiellutin C and its biological evaluation
  35. Enantioselective synthesis of the C5–C23 segment of biselyngbyaside
  36. Synthesis and Self‐Assembly of Bolaamphiphiles Based on β‐Amino Acids or an Alcohol
  37. Synthetic Studies towards Stachybotrin C
  38. A ligand-free copper(II)-catalyzed three-component reaction in poly(ethylene glycol) medium: a versatile protocol for the preparation of selected 3-indole derivatives
  39. Asymmetric Synthesis of the C14–C26 Building Block of Eribulin Mesylate
  40. Synthesis of new 4-methyl-3-piperidones via an iron-catalyzed intramolecular tandem isomerization–aldolisation process
  41. Asymmetric Syntheses of All Stereoisomers of 3-Hydroxyproline; A Constituent of Several Bioactive Compounds
  42. Total Synthesis of Gabosines
  43. ChemInform Abstract: Synthesis of O‐Spiro‐C‐Aryl Glycosides Using Organocatalysis.
  44. Formal synthesis of fumonisin B1, a potent sphingolipid biosynthesis inhibitor
  45. A carbohydrate approach for the formal total synthesis of the prostacyclin analogue (16S)-iloprost
  46. ChemInform Abstract: First Acid Catalyzed Entry to O‐Alkylated Hydroximides from Benzylic Alcohols.
  47. Synthesis of O-Spiro-C-Aryl Glycosides Using Organocatalysis
  48. Synthesis and neurite growth evaluation of new analogues of honokiol, a neolignan with potent neurotrophic activity
  49. Formal synthesis of (+)-didemniserinolipid B
  50. aza-Flavanones as potent cross-species microRNA inhibitors that arrest cell cycle
  51. An improved synthesis of lysosomal activated mustard prodrug for tumor-specific activation and its cytotoxic evaluation
  52. Formal Synthesis of Antiplatelet Drug, Beraprost
  53. Total synthesis of gabosines via an iron-catalyzed intramolecular tandem aldol process
  54. ChemInform Abstract: A Chiral Pyrrolidine‐Pyrazole Catalyst for the Enantioselective Michael Addition of Carbonyls to Nitroolefins.
  55. First Acid‐Catalyzed Entry to O‐Alkylated Hydroximides from Benzylic Alcohols
  56. Synthesis of the ‘southern’ tripeptide of Cyclomarins A and C having novel anti-tuberculocidal mode of action
  57. ChemInform Abstract: Click Reaction on in situ Generated β‐Azidostyrenes from Cinnamic Acid Using CAN—NaN3: Synthesis of N‐Styryl Triazoles.
  58. Click reaction on in situ generated β-azidostyrenes from cinnamic acid using CAN–NaN3: synthesis of N-styryl triazoles
  59. Practical Syntheses of (2S)‐R207910 and (2R)‐R207910 (Eur. J. Org. Chem. 11/2011)
  60. ChemInform Abstract: Hydroxyphthalimide Allied Triazole‐Pyrrolidine Catalyst for Asymmetric Michael Additions in Water.
  61. Practical Syntheses of (2S)‐R207910 and (2R)‐R207910
  62. A chiral pyrrolidine-pyrazole catalyst for the enantioselective Michael addition of carbonyls to nitroolefins
  63. Intramolecular copper(I)-catalyzed 1,3-dipolar cycloaddition of azido-alkynes: synthesis of triazolo-benzoxazepine derivatives and their biological evaluation
  64. Stereoselective Synthesis of Tetrahydropyranyl Diarylheptanoids (-)-Centrolobine and (+)-Centrolobine
  65. Hydroxyphthalimide allied triazole-pyrrolidine catalyst for asymmetric Michael additions in water
  66. Synthesis of Readily Accessible Triazole-Linked Dimer Deoxynucleoside Phosphoramidite for Solid-Phase Oligonucleotide Synthesis
  67. ChemInform Abstract: The First Synthesis of 2‐Amino‐1,4‐dihydroquinolines.
  68. ChemInform Abstract: Proline—Threonine Dipeptide as an Organocatalyst for the Direct Asymmetric Aldol Reaction.
  69. Novel helical foldamers: organized heterogeneous backbone folding in 1 : 1 α/nucleoside-derived-β-amino acid sequences
  70. ChemInform Abstract: From Vinyl Pyranoses to Carbasugars by an Iron-Catalyzed Reaction Complementary to Classical Ferrier Carbocyclization.
  71. ChemInform Abstract: Enantiopure Cycloalkane Fused Tetrahydropyrans Through Domino Michael—Ketalizations with Organocatalysis.
  72. Total Synthesis of Bengazole A
  73. The first synthesis of 2-amino-1,4-dihydroquinolines
  74. Toward Tubulysin: Gram-Scale Synthesis of Tubuvaline-Tubuphenylalanine Fragment
  75. Backbone Regulation Mimicry by β‐Peptidic Foldamers: Formation of a 10‐Helix in a Mixed 6‐Strand/14‐Helix Conformational Pool
  76. Synthesis of the C10–C24 fragment of (+)-cannabisativine
  77. Proline–threonine dipeptide as an organocatalyst for the direct asymmetric aldol reaction
  78. From vinyl pyranoses to carbasugars by an iron-catalyzed reaction complementary to classical Ferrier carbocyclization
  79. Enantiopure cycloalkane fused tetrahydropyrans through domino Michael–ketalizations with organocatalysis
  80. β-Strand mimetics: formation of bend-strands in oligomers of enantiomeric β-amino acids
  81. Total Synthesis of Azumamide E and Sugar Amino Acid-Containing Analogue
  82. β-Sugar Aminoxy Peptides As Rigid Secondary Structural Scaffolds
  83. An efficient process for the resolution of cis-4-O-protected-2-cyclopenten-1,4-diol using pancreatin lipase in [C8mim][PF6] as a reusable system
  84. ChemInform Abstract: Tris(pentafluorophenyl)borane-Catalyzed Three-Component Reaction for the Synthesis of 1,8-Dioxodecahydroacridines under Solvent-Free Conditions.
  85. Total Synthesis of Hyacinthacine A1, a Glycosidase Inhibitor
  86. Spirastrellolide B: The Synthesis of Southern (C9−C25) Region
  87. Asymmetric Synthesis of (-)-6-epi-Centrolobine
  88. Synthesis and Conformational Studies of a Hybrid Cyclic Peptide Based on cis - β -Furanoid Sugar Amino Acid (FSAA) and Ornithine
  89. Tris(pentafluorophenyl)borane-Catalyzed Three-Component Reaction for the Synthesis of 1,8-Dioxodecahydroacridines under Solvent-Free Conditions
  90. ChemInform Abstract: Applications of Zirconium(IV) Chloride in Organic Synthesis
  91. Applications of Zirconium(IV) Chloride in Organic Synthesis
  92. ChemInform Abstract: Stereoselective Formal Total Synthesis of the Cyclodepsipeptide (‐)‐Spongidepsin (I).
  93. Ionic Liquids as Recyclable Solvents for Diethylaminosulfur Trifluoride (DAST) Mediated Fluorination of Alcohols and Carbonyl Compounds.
  94. Recent Developments in the Synthesis of Prostaglandins and Analogues
  95. Stereoselective formal total synthesis of the cyclodepsipeptide (−)-spongidepsin
  96. Palladium‐Catalyzed Reduction of N‐(tert‐Butoxycarbonyl)indoles by Polymethylhydrosiloxane.
  97. A Catalytic Method for Converting Vinylic Furanoses into Cyclopentenones
  98. Innentitelbild: A Catalytic Method for Converting Vinylic Furanoses into Cyclopentenones (Angew. Chem. 33/2007)
  99. Inside Cover: A Catalytic Method for Converting Vinylic Furanoses into Cyclopentenones (Angew. Chem. Int. Ed. 33/2007)
  100. Inter and intramolecular copper(I)-catalyzed 1,3-dipolar cycloaddition of azido-alkynes: synthesis of furanotriazole macrocycles
  101. A Catalytic Method for Converting Vinylic Furanoses into Cyclopentenones
  102. Ionic liquids as recyclable solvents for diethylaminosulfur trifluoride (DAST) mediated fluorination of alcohols and carbonyl compounds
  103. Recent Developments in the Synthesis of Prostaglandins and Analogues
  104. Palladium-Catalyzed Reduction of N-(tert-Butoxycarbonyl)indoles by Polymethylhydrosiloxane
  105. Formation of left-handed helices in hybrid peptide oligomers with cis β-sugar amino acid and l-Ala as building blocks
  106. Stereoselective synthesis of (−)-bulgecinine hydrochloride and its C-2 epimer from l-ascorbic acid
  107. Practical and Highly Stereoselective Approaches to the Total Synthesis of (‐)‐Codonopsinine.
  108. A Facile and Chemoselective Conjugate Reduction Using Polymethylhydrosiloxane (PMHS) and Catalytic B(C6F5)3.
  109. Tris(pentafluorophenyl)borane-Catalyzed Synthesis of N-Benzyl Pyrrolidines
  110. Copper‐Catalyzed N‐Arylation of Amines/Amides in Poly(ethylene glycol) as Recyclable Solvent Medium.
  111. Polyethylene Glycol 400 as Superior Solvent Medium Against Ionic Liquids for Catalytic Hydrogenations with PtO2.
  112. Practical and highly stereoselective approaches to the total synthesis of (−)-codonopsinine
  113. Poly(ethylene Glycol) (400) as Superior Solvent Medium against Ionic Liquids for Catalytic Hydrogenations with PtO2
  114. Copper-Catalyzed N-Arylation of Amines/Amides in Poly(ethylene glycol) as Recyclable Solvent Medium
  115. Oligomers of cis-β-norbornene amino acid: Formation of β-strand mimetics
  116. Self-assembly of cyclic homo- and hetero-β-peptides with cis- furanoid sugar amino acid and β-hGly as building blocks
  117. A facile and chemoselective conjugate reduction using polymethylhydrosiloxane (PMHS) and catalytic B(C6F5)3
  118. Palladium‐Triethylborane‐Triggered Direct and Regioselective Conversion of Allylic Alcohols to Allyl Phenyl Sulfones.
  119. The first simple and efficient synthesis of the unusual dipeptide part of Phomopsin A
  120. Palladium−Triethylborane-Triggered Direct and Regioselective Conversion of Allylic Alcohols to Allyl Phenyl Sulfones
  121. Synthesis of Fluoro Analogues of Unsaturated Fatty Acids and Corresponding Acyclic Metabolites
  122. Expanding the Conformational Pool of cis-β-Sugar Amino Acid:  Accommodation of β-hGly Motif in Robust 14-Helix
  123. Synthesis of Fluoro Analogues of Unsaturated Fatty Acids and Corresponding Acyclic Metabolites
  124. Formation of a Stable 14-Helix in Short Oligomers of Furanoid cis-β-Sugar-Amino Acid
  125. Stetter Reaction in Room Temperature Ionic Liquids and Application to the Synthesis of Haloperidol
  126. Applications of Trivalent and Pentavalent Tantalum in Organic Synthesis
  127. Synthesis and Preliminary Use of Novel Acrylic Ester‐Derived Task‐Specific Ionic Liquids.
  128. Synthesis and preliminary use of novel acrylic ester-derived task-specific ionic liquids
  129. Natural Product Hybrids as New Leads for Drug Discovery
  130. Naturstoffhybride als neue Leitstrukturen bei der Wirkstoffsuche
  131. Natural Product Hybrids as New Leads for Drug Discovery
  132. Soluble Polymer Supported Asymmetric Synthesis (SPSAS)
  133. Study of Bamford-Stevens Reaction onα-Oxy Tosylhydrazones