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  1. A Critical Review on Therapeutic Potential of Benzimidazole Derivatives: A Privileged Scaffold

    Article • Medicinal Chemistry, March 2024, Bentham Science Publishers

    Prabakaran A, Dr Afzal Basha Shaik

  2. Antitubercular activity assessment of fluorinated chalcones, 2-aminopyridine-3-carbonitrile and 2-amino-4H-pyran-3-carbonitrile derivatives: In vitro, molecular docking and in-silico drug likeliness studies

    Article • PLoS ONE, June 2022, PLOS

    Dr Afzal Basha Shaik

  3. Antitubercular and antioxidant activities of hydroxy and chloro substituted chalcone analogues: Synthesis, biological and computational studies

    Article • Arabian Journal of Chemistry, February 2022, Elsevier

    Dr Afzal Basha Shaik

  4. Forging of nicotine for the effective management of diabetic wounds: A hybrid of scaffold hopping and molecular dynamics simulation approaches

    Article • Arabian Journal of Chemistry, February 2022, Elsevier

    Dr Afzal Basha Shaik

  5. Heterogeneous graphitic carbon nitrides in visible-light-initiated organic transformations

    Article • Green Chemistry, January 2022, Royal Society of Chemistry

    Dr Afzal Basha Shaik, Dr Girish YR

  6. Ureidosulfocoumarin Derivatives As Selective and Potent Carbonic Anhydrase IX and XII Inhibitors

    Article • ChemMedChem, December 2021, Wiley

    Dr Afzal Basha Shaik

  7. In Silico and In Vitro Studies for Benzimidazole Anthelmintics Repurposing as VEGFR-2 Antagonists: Novel Mebendazole-Loaded Mixed Micelles with Enhanced Dissolution and Anticancer Activity

    Article • ACS Omega, December 2021, American Chemical Society (ACS)

    Dr Afzal Basha Shaik

  8. Assessment of the Antimicrobial and Antiproliferative Activities of Chloropyrazine-Tethered Pyrimidine Derivatives: In Vitro, Molecular Docking, and In-Silico Drug-Likeness Studies

    Article • Applied Sciences, November 2021, MDPI AG

    Dr Afzal Basha Shaik

  9. 2D-Quantitative structure activity relationship (QSAR) modeling, docking studies, synthesis and in-vitro evaluation of 1,3,4-thiadiazole tethered coumarin derivatives as antiproliferative agents

    Article • Journal of Saudi Chemical Society, July 2021, Elsevier

    Dr Afzal Basha Shaik

  10. A key review on oxadiazole analogs as potential methicillin-resistant Staphylococcus aureus (MRSA) activity: Structure-activity relationship studies

    Article • European Journal of Medicinal Chemistry, July 2021, Elsevier

    Dr Afzal Basha Shaik

  11. Design, multistep synthesis and in-vitro antimicrobial and antioxidant screening of coumarin clubbed chalcone hybrids through molecular hybridization approach

    Article • Arabian Journal of Chemistry, June 2021, Elsevier

    Dr Afzal Basha Shaik

  12. Thiazole–Chalcone Hybrids as Prospective Antitubercular and Antiproliferative Agents: Design, Synthesis, Biological, Molecular Docking Studies and In Silico ADME Evaluation

    Article • Molecules, May 2021, MDPI AG

    Dr Afzal Basha Shaik

  13. Synthesis, and biological screening of chloropyrazine conjugated benzothiazepine derivatives as potential antimicrobial, antitubercular and cytotoxic agents

    Article • Arabian Journal of Chemistry, February 2021, Elsevier

    Dr Afzal Basha Shaik

  14. Design, Synthesis, and Antibacterial and Antifungal Activities of Novel Trifluoromethyl and Trifluoromethoxy Substituted Chalcone Derivatives

    Article • Pharmaceuticals, November 2020, MDPI AG

    Dr Afzal Basha Shaik

  15. Synthesis, Biological and Computational Evaluation of Novel 2,3-dihydro-2-aryl-4-(4- isobutylphenyl)-1,5-benzothiazepine Derivatives as Anticancer and Anti-EGFR Tyrosine Kinase Agents

    Article • Anti-Cancer Agents in Medicinal Chemistry, August 2020, Bentham Science Publishers

    Dr Afzal Basha Shaik

  16. Design, Facile Synthesis and Characterization of Dichloro Substituted Chalcones and Dihydropyrazole Derivatives for Their Antifungal, Antitubercular and Antiproliferative Activities

    Article • Molecules, July 2020, MDPI AG

    Dr Afzal Basha Shaik

  17. Antimicrobial, Antioxidant, and Anticancer Activities of Some Novel Isoxazole Ring Containing Chalcone and Dihydropyrazole Derivatives

    Article • Molecules, February 2020, MDPI AG

    Dr Afzal Basha Shaik

  18. Synthesis of Novel and Potential Antimicrobial, Antioxidant and Anticancer Chalcones and Dihydropyrazoles Bearing Isoxazole Scaffold

    Article • Proceedings, January 2020, MDPI AG

    Dr Afzal Basha Shaik

  19. Synthesis and screening of novel lipophilic diarylpropeones as prospective antitubercular, antibacterial and antifungal agents

    Article • Biointerface Research in Applied Chemistry, June 2019, AMG Transcend Association

    Dr Afzal Basha Shaik

  20. Novel Pyrimidine Derivatives from 2,5-Dichloro-3-acetylthienyl Chalcones as Antifungal, Antitubercular and Cytotoxic Agents: Design, Synthesis, Biological Activity and Docking Study

    Article • Asian Journal of Chemistry, April 2019, Asian Journal of Chemistry

    Dr Afzal Basha Shaik

  21. Synthesis, characterization and antitubercular evaluation of some new isoxazole appended 1-carboxamido-4,5-dihydro-1H-pyrazoles

    Article • Journal of Research in Pharmacy, February 2019, Marmara University

    Dr Afzal Basha Shaik

  22. SYNTHESIS, ANTIBACTERIAL, ANTIFUNGAL ANTITUBERCULAR ACTIVITIES AND MOLECULAR DOCKING STUDIES OF NITROPHENYL DERIVATIVES

    Article • International Journal of Pharma and Bio Sciences, February 2019, International Journal of Pharma and Bio Sciences

    Dr Afzal Basha Shaik

  23. Synthesis, biological evaluation and molecular docking studies of new pyrazolines as an antitubercular and cytotoxic agents

    Article • Infectious Disorders - Drug Targets, December 2018, Bentham Science Publishers

    Bontha Venkata Subrahmanya Lokesh, Dr Afzal Basha Shaik

  24. (E)-1-(2′,4′-Dimethyl)-(5-acetylthiazole)-(2,4″-difluorophenyl)-prop-2-en-1-one

    Article • Molbank, September 2018, MDPI AG

    Dr Afzal Basha Shaik

  25. Synthesis and Biological Activity of Novel 2,5-Dichloro-3-Acetylthiophene Chalcone Derivatives

    Article • Indian Journal of Pharmaceutical Education and Research, December 2017, EManuscript Services

    Dr Afzal Basha Shaik

  26. BIOLOGICAL EVALUATION OF MERREMIA EMARGINATA FOR ANTIBACTERIAL, ANTIFUNGAL AND ANTIOXIDANT ACTIVITIES

    Article • World Journal of Pharmacy and Pharmaceutical Sciences, July 2017, World Journal of Pharmacy and Pharmaceutical Sciences

    Dr Afzal Basha Shaik

  27. Article • International Journal of Pharmaceutical Sciences and Research, June 2017, International Journal of Pharmaceutical Sciences and Research

    Dr Afzal Basha Shaik

  28. Synthesis, Antimicrobial, and Computational Evaluation of Novel Isobutylchalcones as Antimicrobial Agents

    Article • International Journal of Medicinal Chemistry, January 2017, Hindawi Publishing Corporation

    Dr Afzal Basha Shaik