All Stories

  1. Anti-Migratory Activity of Brazilin Chemodiversification on Breast Cancer Cells
  2. Microwave-Assisted Hydrolysis of Ethyl Azolylacetates and Cinnamates with K2CO3: Synthesis of Potassium Carboxylates
  3. Stereodivergent Synthesis of the Four Stereoisomers of Diethyl 4-Hydroxyphosphopipecolate from Ethyl (R)-4-Cyano-3-hydroxybutanoate
  4. Stereocontrolled Synthesis of Phosphoproline Analogues Containing a trans-Fused Octahydroindole Bicyclic System
  5. A Computational Method for the Binding Mode Prediction of COX-1 and COX-2 Inhibitors: Analyzing the Union of Coxibs, Oxicams, Propionic and Acetic Acids
  6. Stereodivergent Synthesis of rac-cis- and rac-trans-4-Hydroxyphosphopipecolic Acids
  7. First Stereoselective Synthesis of Diethyl cis- and trans-(4-Hydroxy-1,2,3,4-tetrahydroquinolin-2-yl)phosphonates and Ethyl Phenylphosphinates from Quinolin-4(1H)-one
  8. Iodine(III)‐Mediated Electrophilic Chlorination and Catalytic Nitration of N‐Tosyl Anilines
  9. Diastereoselective Phosphonylation of Chiral Cyclic Imines for the Synthesis of Phosphoproline Derivatives
  10. Synthesis of 1,5‐Disubstituted Tetrazole−Indolizine Bis‐Heterocycles and Their Copper (II) Recognizing Properties
  11. An efficient synthesis of cis-4-hydroxyphosphonic and cis-4-hydroxyphosphinic analogs of pipecolic acid from cyclic enaminones
  12. Experimental and theoretical study of novel aminobenzamide–aminonaphthalimide fluorescent dyads with a FRET mechanism
  13. Discovery of Octahydroisoindolone as a Scaffold for the Selective Inhibition of Chitinase B1 from Aspergillus fumigatus: In Silico Drug Design Studies
  14. Stereocontrolled Synthesis of Enantiopure cis-Fused Octahydroisoindolones via Chiral Oxazoloisoindolone Lactams
  15. Versatile optical response of pyridylalkyl naphthalenediimides in the interaction with metal ions
  16. Synthesis of phthalimides, isoindolin-1-ones and isoindolines bearing aminobenzoic acids as a new fluorescent compounds
  17. New approaches towards the synthesis of 1,2,3,4-tetrahydro isoquinoline-3-phosphonic acid (TicP)
  18. Structural Diversity using Hyp “Customizable Units”: Proof‐of‐Concept Synthesis of Sansalvamide‐Related Antitumoral Peptides
  19. Practical synthesis of 3-(2-arylethylidene)isoindolin-1-ones (analogues of AKS-182) and 3-(2-arylethylidene)isobenzofuran-1(3H)-ones
  20. Synthesis, characterization and anion recognition studies of new fluorescent alkyl bis(naphthylureylbenzamide)-based receptors
  21. Stereoselective synthesis of acyclic α,α-disubstituted α-amino acids derivatives from amino acids templates
  22. Practical Synthesis of 1,2,3,4-Tetrahydroisoquinoline-1-phosphonic and -1-phosphinic Acids through Kabachnik–Fields and Aza-Pudovik Reaction
  23. Highly Diastereoselective Synthesis of Cyclic α-Aminophosphonic and α-Aminophosphinic Acids from Glycyl-l -Proline 2,5-Diketopiperazine
  24. A Straightforward Synthesis of Six‐Membered‐Ring Heterocyclic α‐Aminophosphonic Acids from N ‐Acyliminium Ions
  25. 000Synthesis of new α-aminophosphonates: Evaluation as anti-inflammatory agents and QSAR studies
  26. Reactions of Piperazin-2-one, Morpholin-3-one, and Thiomorpholin-3-one with Triethyl Phosphite Prompted by Phosphoryl Chloride: Scope and Limitations
  27. Synthesis and anion recognition studies of new oligomethylene bis(nitrophenylureylbenzamide) receptors
  28. An Efficient Method for the Synthesis of New Non‐Symmetrical Naphthalenediimides
  29. Efficient PhB(OH) 2 -catalyzed one-pot synthesis of 3-substituted isoindolin-1-ones and isobenzofuran-1(3 H )-ones under solvent free conditions
  30. Synthesis, biological activity and molecular modelling studies of shikimic acid derivatives as inhibitors of the shikimate dehydrogenase enzyme of Escherichia coli
  31. First and Highly Stereoselective Synthesis of Both Enantiomers of Octahydroindole-2-phosphonic Acid (OicP)
  32. First practical synthesis of novel 1-phosphonylated pyrrolo[1,2-a ]pyrazine derivatives
  33. Synthesis and anion recognition studies of new ureylbenzamide-based receptors
  34. Stereoselective Synthesis of α‐Aminophosphonic Acids through Pudovik and Kabachnik‐Fields Reaction
  35. Synthesis, antimycobacterial and cytotoxic activity of α,β-unsaturated amides and 2,4-disubstituted oxazoline derivatives
  36. ChemInform Abstract: An Update on the Stereoselective Synthesis of γ-Amino Acids
  37. An update on the stereoselective synthesis of γ-amino acids
  38. Stereoselective Synthesis of α-Amino-H-phosphinic Acids and Derivatives
  39. ChemInform Abstract: First Synthesis of (R)- and (S)-1,2,3,4-Tetrahydroisoquinoline-3-phosphonic Acid (TicP) Using a Pictet-Spengler Reaction.
  40. Practical and Efficient Synthesis of α-Aminophosphonic Acids Containing 1,2,3,4-Tetrahydroquinoline or 1,2,3,4-Tetrahydroisoquinoline Heterocycles
  41. Stereoselective Synthesis of α-Amino-C-phosphinic Acids and Derivatives
  42. ChemInform Abstract: Convenient Synthesis of Cyclic α-Aminophosphonates by Alkylation-Cyclization Reaction of Iminophosphoglycinates Using Phase-Transfer Catalysis.
  43. First Synthesis of (R)- and (S)-1,2,3,4-Tetrahydroisoquinoline-3-phosphonic Acid (TicP) Using a Pictet-Spengler Reaction
  44. Novel naphthalimide–aminobenzamide dyads asOFF/ONfluorescent supramolecular receptors in metal ion binding
  45. Practical synthesis of novel phosphonopeptides containing AibP
  46. Efficient Synthesis of β-Aryl-γ-lactams and Their Resolution with (S)-Naproxen: Preparation of (R)- and (S)-Baclofen
  47. Convenient Synthesis of Cyclic α-Aminophosphonates by Alkylation-Cyclization Reaction of Iminophosphoglycinates Using Phase-Transfer Catalysis
  48. Synthesis of Chiral 1,4,2-Oxazaphosphepines
  49. ChemInform Abstract: First Practical and Efficient Synthesis of 3-Phosphorylated β-Carboline Derivatives Using the Pictet-Spengler Reaction.
  50. ChemInform Abstract: Synthesis of β-Hydroxyacetamides from Unactivated Ethyl Acetates under Base-Free Conditions and Microwave Irradiation.
  51. ChemInform Abstract: An Update on the Stereoselective Synthesis of α-Aminophosphonic Acids and Derivatives
  52. Synthesis and Characterization ofm-Terphenyl (1,3-Diphenylbenzene) Compounds Containing Trifluoromethyl Groups
  53. An update on the stereoselective synthesis of α-aminophosphonic acids and derivatives
  54. First Practical and Efficient Synthesis of 3-Phosphorylated β-Carboline Derivatives Using the Pictet-Spengler Reaction
  55. Synthesis of β-hydroxyacetamides from unactivated ethyl acetates under base-free conditions and microwave irradiation
  56. ChemInform Abstract: Phenylphosphonic Acid as Efficient and Recyclable Catalyst in the Synthesis of α-Aminophosphonates under Solvent-Free Conditions.
  57. ChemInform Abstract: Synthesis of 3-Alkylideneisoindolinones and Isoindolones by a Horner-Wadsworth-Emmons Reaction.
  58. ChemInform Abstract: Diastereoselective Synthesis of Novel 5-Substituted Morpholine-3-phosphonic Acids: Further Exploitation of N-Acyliminium Intermediates.
  59. ChemInform Abstract: Practical and Efficient Synthesis of Chiral 2,4-Disubstituted Oxazolines from β-Phosphonoamides.
  60. Phenylphosphonic Acid as Efficient and Recyclable Catalyst in the Synthesis of α-Aminophosphonates under Solvent-Free Conditions
  61. Diastereoselective synthesis of novel 5-substituted morpholine-3-phosphonic acids: further exploitation of N-acyliminium intermediates
  62. Synthesis of 3-alkylideneisoindolinones and isoindolones by a Horner–Wadsworth–Emmons reaction
  63. Practical and efficient synthesis of chiral 2,4-disubstituted oxazolines from β-phosphonoamides
  64. A Novel and Highly Regioselective Synthesis of New Carbamoylcarboxylic Acids from Dianhydrides
  65. A versatile synthesis of bicyclic lactams from 1,8-naphthalaldehydic acid: an extension of Meyers’ method
  66. ChemInform Abstract: Practical and Highly Stereoselective Synthesis of 3-(Arylmethylene)isoindolin-1-ones from 2-Formylbenzoic Acid.
  67. ChemInform Abstract: Synthesis of Quaternary α-Aminophosphonic Acids
  68. ChemInform Abstract: Phenylboronic Acid as Efficient and Eco-Friendly Catalyst for the One-Pot, Three-Component Synthesis of α-Aminophosphonates under Solvent-Free Conditions.
  69. Practical and high stereoselective synthesis of 3-(arylmethylene)isoindolin-1-ones from 2-formylbenzoic acid
  70. ChemInform Abstract: Stereoselective Synthesis of α-Aminophosphonic Acid Analogues of the 20 Proteinogenic α-Amino Acids
  71. Synthesis of quaternary α-aminophosphonic acids
  72. Phenylboronic Acid as Efficient and Eco-Friendly Catalyst for the One-Pot, Three-Component Synthesis of α-Aminophosphonates under Solvent-Free Conditions
  73. ChemInform Abstract: An Easy Approach for the Synthesis of N-Substituted Isoindolin-1-ones.
  74. Stereoselective Synthesis of α-Aminophosphonic Acids Analogs of the 20 Proteinogenic α-Amino Acids
  75. An Easy Approach for the Synthesis of N-Substituted Isoindolin-1-ones
  76. Synthesis of cis- and trans-3-Aminocyclohexanols by Reduction of β-Enaminoketones
  77. Microwave-Assisted Improved Synthesis of Oxazolidin-2-ones, Oxazolidine-2-thiones and Thiazolidine-2-thione Chiral Auxiliaries
  78. Synthesis of Phosphoproline Derivatives with an Octahydroisoindole Structure
  79. One-pot three-component highly diastereoselective synthesis of isoindolin-1-one-3-phosphonates under solvent and catalyst free-conditions
  80. Stereodivergent Synthesis of Two Novel α-Aminophosphonic Acids Characterised by a cis-Fused Octahydroindole System
  81. First Total Synthesis of 5-Hydroxy-3-methyl-4-propylsulfanyl-5H-furan-2-one: A Cancer Chemopreventive Agent
  82. Reversal Diastereoselectivity in the Benzylation of Phosphonopropanoamides
  83. ChemInform Abstract: Uncatalyzed One-Pot Diastereoselective Synthesis of α-Amino Phosphonates under Solvent-Free Conditions.
  84. Study of the fragmentation pathway of α-aminophosphonates by chemical ionization and fast atom bombardment mass spectrometry
  85. Uncatalyzed One-Pot Diastereoselective Synthesis of α-Amino Phosphonates Under Solvent-Free Conditions
  86. ChemInform Abstract: Enantioselective Diels-Alder Reactions Catalyzed by Chiral Magnesium Lewis Acids Prepared from Hydroxysulfoxides.
  87. ChemInform Abstract: Synthesis of Aldehydes from Oxiranes Using Silica Gel as Reagent.
  88. ChemInform Abstract: Improved Large Scale Preparation of Both Enantiomers of Methyl p-Tolyl Sulfoxide from Diacetone-D-glucose.
  89. ChemInform Abstract: A Convenient Synthesis of (E)-γ-Hydroxy- and (E)-γ-Keto-. alpha.,β-Unsaturated Sulfoxides.
  90. Stereochemistry of base-induced cleavage of methoxide ion on cis- and trans-1,4-diphenylphosphorinanium salts. A different behavior with a phenyl substituent
  91. ChemInform Abstract: Conformational Preference of the Sulfinyl Group in Six-Membered Heterocycles
  92. ChemInform Abstract: Stereoselective Synthesis of GABOB, Carnitine and Statine Phosphonates Analogues.
  93. ChemInform Abstract: Palladium-Catalyzed Allylic Nucleophilic Substitution Reactions of (E)-γ-Acetoxy-α,β-unsaturated p-Tolylsulfoxides.
  94. ChemInform Abstract: Diastereoselective Reduction of β-Ketophosphonates Derived from Amino Acids. A New Entry to Enantiopure β-Hydroxy-γ-aminophosphonate Derivatives.
  95. Synthesis of syn-γ-Amino-β-hydroxyphosphonates by Reduction of β-Ketophosphonates Derived from L-Proline and L-Serine
  96. Stereoselective synthesis of GABOB, carnitine and statine phosphonates analogues
  97. ChemInform Abstract: Recent Progress on the Stereoselective Synthesis of Cyclic Quaternary α-Amino Acids.
  98. ChemInform Abstract: Stereoselective Synthesis of α-Aminophosphonic Acids and Derivatives.
  99. Recent progress on the stereoselective synthesis of cyclic quaternary α-amino acids
  100. An overview of stereoselective synthesis of α-aminophosphonic acids and derivatives
  101. Reversal of diastereoselectivity in the benzylation of the lithium enolates of phosphonopropanoamides by changing the base equivalents
  102. ChemInform Abstract: A Convenient Method for the Preparation of Chiral Phosphonoacetamides and Their Horner-Wadsworth-Emmons Reaction.
  103. A practical synthesis of syn- and anti-α,β-dihydroxyphosphinates via diastereoselective reduction of α-phosphinoyl ketones
  104. A convenient method for the preparation of chiral phosphonoacetamides and their Horner–Wadsworth–Emmons reaction
  105. Stereoselective Synthesis of γ-Amino Acids
  106. Stereoselective synthesis of γ-amino acids
  107. Preparation of dimethyl (R)- and (S)-2-(2-hydroxyphenyl)-2-hydroxyethylphosphonate derived from salicylaldehyde via resolution using (S)-methoxyphenylacetic acid (MPA)
  108. Practical and Efficient Synthesis of (E)-α,β-Unsaturated Amides Bearing (S)-α-Methylbenzylamine from 2-Phosphonamides via Horner—Wadsworth—Emmons Reaction.
  109. Practical and Efficient Synthesis of (E)-α,β-Unsaturated Amides Bearing (S)-α-Methylbenzylamine from 2-Phosphonamides via Horner-Wadsworth-Emmons Reaction
  110. Synthesis of some monocyclic analogues of mycophenolic acid via the Johnson ortho ester Claisen rearrangement
  111. Synthesis of New 1,3-Oxaphosphorinanium Salts. Stereochemistry of Hydroxide-Induced Displacement of Methoxide Ion
  112. Asymmetric Alkylation of Dimethoxyphosphoryl-N-[1-(S)-α-methylbenzyl]acetamide Enolates. Synthesis of Both Stereoisomers from the Same Source of Chirality by Changing the Equivalents of LDA.
  113. Preparation of phosphostatine and phosphoepistatine from L-leucine via high diastereoselective reduction of 3-amino-2-ketophosphonates
  114. Diastereoselective Reduction of Dimethyl ?-[(N-p-Toluenesulfonyl)amino]-?-ketophosphonates Derived from Amino Acids.
  115. Asymmetric alkylation of dimethoxyphosphoryl-N-[1-(S)-α-methylbenzyl]acetamide enolates. Synthesis of both stereoisomers from the same source of chirality by changing the equivalents of LDA
  116. Diastereoselective reduction of dimethyl γ-[(N-p-toluenesulfonyl)amino]-β-ketophosphonates derived from amino acids
  117. Highly diastereoselective reduction of β-ketophosphonates bearing homochiral bis(α-methylbenzyl)amine: preparation of both enantiomers of phosphogabob (GABOBP)
  118. Highly Diastereoselective Synthesis of anti-γ-N-Benzylamino-β-hydroxyphosphonates.
  119. Preparation of dimethyl (R)- and (S)-2-(2-aminophenyl)-2-hydroxyethylphosphonate from anthranilic acid
  120. Highly Diastereoselective Addition of Et2AlCN to β-Keto Amides Derived from (S)-4-Isopropyl-2-oxazolidinone.
  121. Highly diastereoselective synthesis of anti-γ-N-benzylamino-β-hydroxyphosphonates
  122. Diels–Alder reaction of optically active (E)-γ-keto-α,β-unsaturated p-tolylsulfoxides with cyclopentadiene
  123. Generation of alkoxyalkynylketenes from a bicyclic precursor. Cycloaddition chemistry with alkynes and theoretical studies regarding the formation of five- versus six-membered ring products
  124. Highly diastereoselective addition of Et2AlCN to β-keto amides derived from (S)-4-isopropyl-2-oxazolidinone
  125. Preparation of (R)- and (S)-γ-amino-β-hydroxypropylphosphonic acid from glycine
  126. Allylic strain effects on the stereochemistry of the alkylation reaction of mycophenolic acid chiral enolates
  127. Diastereoselective reduction of β-ketophosphonates derived from amino acids. A new entry to enantiopure β-hydroxy-γ-aminophosphonate derivatives
  128. Asymmetric synthesis of both diastereomers of protected S-methyl-l-cysteine and S-n-propyl-l-cysteine sulphoxides
  129. Palladium-catalyzed allylic nucleophilic substitution reactions of (E)-γ-acetoxy-α,β-unsaturated p-tolylsulfoxides
  130. ChemInform Abstract: Efficient Preparation of Enantiomerically Pure (E)-γ-Hydroxy-α,β-Unsaturated p-Tolylsulfoxides Using Lipase-Mediated Acylations.
  131. Efficient preparation of enantiomerically pure (E)-γ-hydroxy-α,β-unsaturated p-tolylsulfoxides using lipase-mediated acylations
  132. Conformational Energy of the (η5-Cyclopentadienyl) Iron(II) Dicarbonyl Group
  133. Conformational analysis of 2-(diphenylphosphinoyl)-tetrahydrothiopyran: Lack of additivity of the S-C-P anomeric effect
  134. Chapter 3 Conformational preference of the sulfinyl group in six-membered heterocycles
  135. Enantioselective Diels-Alder reactions catalyzed by chiral magnesium lewis acids prepared from hydroxysulfoxides
  136. Synthesis of Aldehydes from Oxiranes using Silica Gel as Reagent
  137. Improved Large Scale Preparation on Both Enantiomers of Methyl p-Tolyl Sulfoxide from Diacetone-D-glucose
  138. A convenient synthesis of (E)-γ-hydroxy- and (E)-γ-keto-α,β-unsaturated sulfoxides
  139. Conformational analysis of 2-halotetrahydrothiopyran S-oxides. Diminution of the anomeric effect in S(O)-C-X compared to S-C-X segments.
  140. Lack of manifestation of an anomeric effect in 2-diphenylphosphinoyl-1, 3-dioxane and 2-diphenylphosphinoyl-1, 3-oxathiane1
  141. ChemInform Abstract: Synthesis of 4-Hydroxy-4-(2-thienyl)pentamide.
  142. SYNTHESIS OF 4-HYDROXY-4-(2-THIENYL)PENTAMIDE